SCHEMBL28298511

SCHEMBL28298511

CN1CC(c2cc(F)cc(F)c2)CC1=O.NC=S

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 13/20 0.51
PDE4A P27815 3/20 0.47
PDE4B Q07343 1/20 0.47
PDE4C Q08493 1/20 0.47
PDE4D Q08499 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10756940 0.76 BRD4 (0.70) BRD4PDE4APDE4BPDE4CPDE4D
SCHEMBL28296842 0.72 NPC1 (0.37)
SCHEMBL25746011 0.71 BRD4 (0.53) BRD4PDE4APDE4BPDE4CPDE4D
SCHEMBL28288944 0.71 BRD4 (0.49) BRD4PDE4APDE4BPDE4CPDE4D
SCHEMBL24007585 0.70 BRD4 (0.51) BRD4PDE4APDE4BPDE4CPDE4D
SCHEMBL19995938 0.70 MEN1 (0.41) BRD4PDE4APDE4BPDE4CPDE4D
SCHEMBL19996130 0.70 MEN1 (0.41) BRD4PDE4APDE4BPDE4CPDE4D
SCHEMBL19039741 0.70 BRD4 (0.52) BRD4PDE4APDE4BPDE4CPDE4D
SCHEMBL30912528 0.69 BRD4 (0.70) BRD4PDE4APDE4BPDE4CPDE4D
SCHEMBL30912553 0.69 BRD4 (0.70) BRD4PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109715155-A blood brain barrier-penetrating agent dopamine- β -hydroxylase inhibitors 巴尔-波特拉及康邦亚股份有限公司 2019-05-03 CN disclosed