SCHEMBL28298920

SCHEMBL28298920

O=C(CCCCc1ccc(OCc2ccc3ccccc3n2)cc1)Oc1ccc(OCc2ccc3ccccc3n2)cc1

nearest known ligand 0.79

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYSLTR1 Q9Y271 13/20 0.79
CYSLTR2 Q9NS75 9/20 0.79
FFAR1 O14842 1/20 0.69
AKR1B1 P15121 1/20 0.69
GPBAR1 Q8TDU6 1/20 0.58
ALOX5 P09917 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8646512 0.88 CYSLTR1 (1.00) CYSLTR1CYSLTR2FFAR1AKR1B1GPBAR1
SCHEMBL14021512 0.88 CYSLTR1 (0.80) CYSLTR1CYSLTR2FFAR1AKR1B1GPBAR1
SCHEMBL8650454 0.86 CYSLTR1 (0.79) CYSLTR1CYSLTR2FFAR1AKR1B1GPBAR1
SCHEMBL10446560 0.84 CYSLTR1 (0.79) CYSLTR1CYSLTR2FFAR1AKR1B1GPBAR1
SCHEMBL8712492 0.84 CYSLTR1 (0.75) CYSLTR1CYSLTR2FFAR1AKR1B1GPBAR1
SCHEMBL8834916 0.83 FFAR1 (0.83) CYSLTR1CYSLTR2FFAR1AKR1B1GPBAR1
SCHEMBL8709593 0.82 FFAR1 (0.81) CYSLTR1CYSLTR2FFAR1AKR1B1GPBAR1
SCHEMBL8666314 0.82 CYSLTR1 (0.72) CYSLTR1CYSLTR2FFAR1AKR1B1GPBAR1
SCHEMBL9150476 0.82 CYSLTR1 (0.72) CYSLTR1CYSLTR2FFAR1AKR1B1GPBAR1
SCHEMBL10446852 0.81 CYSLTR1 (0.75) CYSLTR1CYSLTR2FFAR1AKR1B1GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109789150-A It is certain to be used to treat bronchiectasic (2S)-N- [(1S) -1- cyano -2- phenethyl] -1,4- oxazepine cycloheptane -2- formamide 英斯梅德股份有限公司 2019-05-21 CN disclosed