SCHEMBL28301245

SCHEMBL28301245

Cc1cc(Nc2nc(C(=O)c3ccccc3)nc3ccccc23)n[nH]1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AURKA O14965 14/20 1.00
AURKB Q96GD4 8/20 1.00
GSK3B P49841 8/20 0.65
SRC P12931 7/20 0.65
EIF2AK2 P19525 1/20 0.65
GSK3A P49840 1/20 0.65
AURKC Q9UQB9 1/20 0.56
NTRK1 P04629 2/20 0.55
JAK2 O60674 3/20 0.55
CYP3A4 P08684 3/20 0.55
CYP2C8 P10632 3/20 0.55
CYP2C9 P11712 3/20 0.55
JAK1 P23458 3/20 0.55
TYK2 P29597 3/20 0.55
CYP2C19 P33261 3/20 0.55
JAK3 P52333 3/20 0.55
ADORA3 P0DMS8 2/20 0.55
CYP1A2 P05177 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL173501 0.93 AURKA (0.88) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL174480 0.92 AURKA (0.84) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL174477 0.88 AURKA (0.79) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL174554 0.87 AURKA (0.76) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL174487 0.86 AURKA (0.74) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL173666 0.85 AURKA (0.73) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL174645 0.84 AURKA (0.72) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL160645 0.83 AURKA (0.71) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL174414 0.83 AURKA (0.73) AURKAAURKBGSK3BSRCEIF2AK2
SCHEMBL174382 0.83 AURKA (0.71) AURKAAURKBGSK3BSRCEIF2AK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106957303-B Quinazoline derivant of selective Aurora A kinase inhibiting activity and preparation method thereof and application 中山大学 2019-06-04 CN disclosed