SCHEMBL28301615

SCHEMBL28301615

C[CH]c1ccc(N(C)C)nc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.53
MAOB P27338 2/20 0.41
APP P05067 6/20 0.38
GRM5 P41594 1/20 0.37
KDM1A O60341 1/20 0.36
MAP3K11 Q16584 1/20 0.35
GBA1 P04062 1/20 0.34
TDO2 P48775 1/20 0.33
HSD17B3 P37058 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30592797 0.81 KCNH2 (0.51) KCNH2MAOBAPPGRM5KDM1A
SCHEMBL934755 0.81 KCNH2 (0.51) KCNH2MAOBAPPGRM5KDM1A
SCHEMBL3664684 0.81 KCNH2 (0.51) KCNH2MAOBAPPGRM5KDM1A
SCHEMBL22198155 0.79 KCNH2 (0.50) KCNH2MAOBAPPGRM5KDM1A
SCHEMBL17081152 0.76 KCNH2 (0.59) KCNH2MAOBAPPGRM5MAPT
SCHEMBL9000457 0.76 KCNH2 (0.59) KCNH2MAOBAPPGRM5KDM1A
SCHEMBL20241361 0.76 KCNH2 (0.47) KCNH2MAOBMAP3K11MAPT
SCHEMBL20241362 0.76 KCNH2 (0.47) KCNH2MAOBMAP3K11MAPT
SCHEMBL23751551 0.75 KCNH2 (0.54) KCNH2MAOBAPPGRM5MAPT
SCHEMBL17081899 0.75 KCNH2 (0.58) KCNH2MAOBAPPGRM5KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109790160-A Pyrido 5-membered aromatic cyclics, preparation method and the usage 上海海和药物研究开发有限公司 2019-05-21 CN disclosed