SCHEMBL2831073

SCHEMBL2831073

CCc1ccc(C#Cc2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.59
APP P05067 1/20 0.57
FFAR1 O14842 6/20 0.55
CYP2A6 P11509 1/20 0.54
FFAR4 Q5NUL3 1/20 0.52
MAPT P10636 1/20 0.50
ASIC3 Q9UHC3 1/20 0.48
KCNH2 Q12809 2/20 0.48
ACACB O00763 1/20 0.46
NPC1 O15118 1/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CHRNB2 P17787 1/20 0.44
CHRNB4 P30926 1/20 0.44
CHRNA3 P32297 1/20 0.44
CHRNA7 P36544 1/20 0.44
CHRNA4 P43681 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5050178 0.90 CYP2A6 (0.64) TP53APPFFAR1CYP2A6ACACB
SCHEMBL8228398 0.90 CYP2A6 (0.64) TP53APPFFAR1CYP2A6ACACB
SCHEMBL9509240 0.83 CYP2A6 (0.56) TP53FFAR1CYP2A6FFAR4ACACB
SCHEMBL7503092 0.83 FFAR1 (0.57) TP53FFAR1CYP2A6FFAR4MAPT
SCHEMBL2833040 0.82 FFAR1 (0.58) APPFFAR1FFAR4MAPTASIC3
SCHEMBL9333011 0.81 CYP2A6 (0.54) TP53APPFFAR1CYP2A6ACACB
SCHEMBL9328231 0.81 CYP2A6 (0.54) TP53FFAR1CYP2A6MAPTKCNH2
SCHEMBL7503100 0.81 CYP2A6 (0.54) TP53FFAR1CYP2A6MAPTKCNH2
SCHEMBL27874223 0.80 TP53 (0.52) TP53APPFFAR1CYP2A6ASIC3
SCHEMBL6734125 0.80 CYP2A6 (0.58) TP53CYP2A6ACACBSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104263380-B A kind of liquid-crystal compounds with high birefringence rate and wide nematic phase temperature range and combinations thereof thing 西安近代化学研究所 2016-08-17 CN disclosed
CN-104263380-A Liquid crystal compound with high birefringence and wide nematic phase temperature interval and composition comprising liquid crystal compound XIAN MODERN CHEMISTRY RES INST 2015-01-07 CN disclosed
EP-1388538-B1 Polymerisation Initiator MERCK PATENT GMBH (DE) 2010-09-01 EP disclosed
US-7728014-B2 Heteroaromatic compounds having sphingosine-1-phosphate (S1P) receptor agonist biological activity ALLERGAN, INC. 2010-06-01 US disclosed
EP-2066633-A1 HETEROAROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR AGONIST AND/OR ANTAGONIST BIOLOGICAL ACTIVITY Allergan, Inc. (US) 2009-06-10 EP disclosed
EP-2064183-A2 HETEROAROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR AGONIST BIOLOGICAL ACTIVITY Allergan, Inc. (US) 2009-06-03 EP disclosed
WO-2008030843-A1 HETEROAROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR AGONIST AND/OR ANTAGONIST BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 2008-03-13 WO disclosed
WO-2008030838-A2 HETEROAROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR AGONIST BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 2008-03-13 WO disclosed
US-20080064872-A1 HETEROAROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR AGONIST BIOLOGICAL ACTIVITY ALLERGAN, INC. 2008-03-13 US disclosed
EP-1388538-A1 Polymerisation Initiator MERCK PATENT GmbH (DE) 2004-02-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080064872-A1 HETEROAROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR AGONIST BIOLOGICAL ACTIVITY S1PR4, S1PR3, S1PR1 TP53 4512/4885APP 1870/4885FFAR1 23/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.