SCHEMBL28357335

SCHEMBL28357335

O=C(Nc1cccc(Cl)c1)c1ccc(C=CC(=O)c2nc3ccccc3[nH]2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.69
MEN1 O00255 5/20 0.69
SMN1; SMN2 Q16637 4/20 0.69
NTSR1 P30989 2/20 0.69
ALDH1A1 P00352 1/20 0.69
PKM P14618 1/20 0.69
HPGD P15428 1/20 0.69
NPY1R P25929 1/20 0.69
NPY2R P49146 1/20 0.69
MAPT P10636 4/20 0.57
RECQL P46063 2/20 0.57
NPSR1 Q6W5P4 2/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
NPC1 O15118 5/20 0.53
RAB9A P51151 4/20 0.53
KDM4E B2RXH2 2/20 0.53
POLB P06746 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28353461 0.89 KMT2A (0.60) KMT2AMEN1SMN1; SMN2NTSR1ALDH1A1
SCHEMBL28883456 0.89 SMN1; SMN2 (0.65) KMT2AMEN1SMN1; SMN2NTSR1ALDH1A1
SCHEMBL28354083 0.88 KMT2A (0.57) KMT2AMEN1SMN1; SMN2NTSR1ALDH1A1
SCHEMBL28353863 0.88 KMT2A (0.66) KMT2AMEN1SMN1; SMN2NTSR1ALDH1A1
SCHEMBL28357255 0.87 KMT2A (0.51) KMT2AMEN1SMN1; SMN2NTSR1ALDH1A1
SCHEMBL28353880 0.86 COMT (0.58) KMT2AMEN1SMN1; SMN2NTSR1ALDH1A1
SCHEMBL28353688 0.86 KMT2A (0.57) KMT2AMEN1SMN1; SMN2NTSR1ALDH1A1
SCHEMBL28357267 0.86 MAPT (0.57) KMT2AMEN1SMN1; SMN2NTSR1ALDH1A1
SCHEMBL28357370 0.83 MEN1 (0.77) KMT2AMEN1SMN1; SMN2NTSR1ALDH1A1
SCHEMBL28353567 0.83 SMN1; SMN2 (0.60) KMT2AMEN1SMN1; SMN2NTSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110615766-A Disubstituted alpha, beta unsaturated ketone, preparation method and application thereof 长治学院 2019-12-27 CN claimed
CN-110615766-B Disubstituted alpha, beta unsaturated ketone, preparation method and application thereof 长治学院 2021-04-20 CN disclosed
CN-110615766-A Disubstituted alpha, beta unsaturated ketone, preparation method and application thereof 长治学院 2019-12-27 CN disclosed