Benzonatate

Benzonatate

SCHEMBL28366

CCCCNc1ccc(C(=O)OCCOCCOCCOCCOCCOCCOCCOCCOCCOC)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 2/20 1.00
CYP3A4 P08684 2/20 1.00
ABCB11 O95342 1/20 1.00
ADRA2B P18089 1/20 1.00
OPRD1 P41143 1/20 1.00
LMNA P02545 4/20 0.67
MAPK1 P28482 3/20 0.67
CYP1A2 P05177 3/20 0.67
MAOA P21397 1/20 0.67
CNR1 P21554 1/20 0.67
DRD4 P21917 1/20 0.67
ACHE P22303 1/20 0.67
HRH2 P25021 1/20 0.67
HTR2A P28223 1/20 0.67
HTR2C P28335 1/20 0.67
NTSR1 P30989 1/20 0.67
HRH1 P35367 1/20 0.67
DRD3 P35462 1/20 0.67
SCN1A P35498 1/20 0.67
HTR2B P41595 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzonatate SCHEMBL14857547 1.00 SCN5A (1.00) SCN5ACYP3A4ABCB11ADRA2BOPRD1
Benzonatate SCHEMBL23646300 0.99 SCN5A (0.97) SCN5ACYP3A4ABCB11ADRA2BOPRD1
Benzonatate SCHEMBL16044570 0.99 SCN5A (0.97) SCN5ACYP3A4ABCB11ADRA2BOPRD1
Benzonatate SCHEMBL23646298 0.99 SCN5A (0.97) SCN5ACYP3A4ABCB11ADRA2BOPRD1
Benzonatate SCHEMBL23646299 0.99 SCN5A (0.97) SCN5ACYP3A4ABCB11ADRA2BOPRD1
Benzonatate SCHEMBL28086694 0.97 SCN5A (0.95) SCN5ACYP3A4ABCB11ADRA2BOPRD1
SCHEMBL14112093 0.96 SCN5A (0.92) SCN5ACYP3A4ABCB11ADRA2BOPRD1
Benzonatate SCHEMBL1375727 0.95 SCN5A (0.91) SCN5ACYP3A4ABCB11ADRA2BOPRD1
Benzonatate SCHEMBL16044024 0.95 SCN5A (0.91) SCN5ACYP3A4ABCB11ADRA2BOPRD1
Benzonatate SCHEMBL16113875 0.93 SCN5A (0.86) SCN5ACYP3A4ABCB11ADRA2BOPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5719 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250319025-A9 COMPOSITIONS COMPRISING MODIFIED PHOSPHOLIPIDS AND USES THEREOF THE CHILDREN'S MEDICAL CENTER CORPORATION (US) 2025-10-16 US claimed
US-20250255781-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-08-14 US claimed
WO-2025150072-A1 A STABLE ORAL PRO-DISPERSION FORMULATION AND IMPLEMENTATIONS THEREOF PULSE PHARMACEUTICALS PVT LTD (IN) 2025-07-17 WO claimed
US-20250205278-A1 METHODS AND COMPOSITIONS FOR WOUND HEALING ABBOTT NICHOLAS L (US) 2025-06-26 US claimed
WO-2025128639-A1 HYDROGELS COMPRISING PROTEIN-STABILIZED NANOPARTICLES FOR EXTENDED RELEASE THE CHILDREN'S MEDICAL CENTER CORPORATION (US) 2025-06-19 WO claimed
WO-2025109556-A1 ROTATOR CUFF SYSTEM ANIKA THERAPEUTICS, INC. (US) 2025-05-30 WO claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
EP-4559410-A1 SURGICAL TOOLS AND SYSTEMS Anika Therapeutics, Inc. (US) 2025-05-28 EP claimed
US-12296043-B2 Liquisoft capsules PATHEON SOFTGELS INC. (US) 2025-05-13 US claimed
WO-2025075976-A2 METHYL-BRANCHED LIPOSOMES FOR SUSTAINED DRUG DELIVERY THE CHILDREN'S MEDICAL CENTER CORPORATION (US) 2025-04-10 WO claimed
EP-0617612-B1 A PROCESS FOR THE PREPARATION OF A SOLID DISPERSION WARNER LAMBERT CO (US) 1997-09-10 EP claimed
CN-1143909-A Antitussive composition containing antitussive and benzydamine ACRAF (IT) 1997-02-26 CN claimed
EP-0748222-A1 ANTITUSSIVE COMPOSITION CONTAINING AN ANTITUSSIVE AND BENZYDAMINE AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.p.A. (IT) 1996-12-18 EP claimed
WO-1996029986-A1 ANTITUSSIVE MICROCAPSULES THE PROCTER & GAMBLE COMPANY (US) 1996-10-03 WO claimed
WO-1995023602-A1 ANTITUSSIVE COMPOSITION CONTAINING AN ANTITUSSIVE AND BENZYDAMINE AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A. (IT) 1995-09-08 WO claimed
EP-0617612-A1 A PROCESS FOR THE PREPARATION OF A SOLID DISPERSION. WARNER LAMBERT CO (US) 1994-10-05 EP claimed
WO-1994018970-A1 COLD/SINUS PREPARATION CONSISTING OF PHENINDAMINE TARTARATE WITH OR WITHOUT THERAPEUTIC AGENTS WARNER-LAMBERT COMPANY (US) 1994-09-01 WO claimed
WO-1993011749-A1 A PROCESS FOR THE PREPARATION OF A SOLID DISPERSION WARNER-LAMBERT COMPANY (US) 1993-06-24 WO claimed
US-4775694-A Antitussive composition BRISTOL-MYERS COMPANY (US) 1988-10-04 US claimed
US-4557934-A ALONG WITH A DIOL PYRROLIDONE OR AN AZACYCLOPENTAN-2-ONE THE PROCTER & GAMBLE COMPANY (US) 1985-12-10 US claimed