SCHEMBL28378486

SCHEMBL28378486

CCCI.O=[N+]([O-])c1ccc2nc[nH]c2c1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.77
NAMPT P43490 1/20 0.77
XDH P47989 1/20 0.77
PARP1 P09874 1/20 0.54
KDM4E B2RXH2 2/20 0.52
RIPK1 Q13546 3/20 0.49
TDP1 Q9NUW8 2/20 0.48
CCNT1 O60563 1/20 0.47
CDK9 P50750 1/20 0.47
NPBWR1 P48145 2/20 0.46
MAPT P10636 4/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
GAA P10253 1/20 0.45
ALDH1A1 P00352 5/20 0.45
LMNA P02545 2/20 0.45
KCNJ1 P48048 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
RAB9A P51151 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alcohol SCHEMBL27894280 0.88 CYP3A4 (0.82) CYP3A4NAMPTXDHPARP1KDM4E
SCHEMBL271341 0.88 CYP3A4 (1.00) CYP3A4NAMPTXDHPARP1KDM4E
SCHEMBL30051508 0.88 CYP3A4 (1.00) CYP3A4NAMPTXDHPARP1KDM4E
SCHEMBL8425549 0.86 CYP3A4 (0.96) CYP3A4NAMPTXDHPARP1KDM4E
Nitric Acid SCHEMBL4907436 0.83 CYP3A4 (0.90) CYP3A4NAMPTXDHPARP1KDM4E
SCHEMBL28832319 0.83 CYP3A4 (0.68) CYP3A4NAMPTXDHPARP1KDM4E
Nitric Acid SCHEMBL11709810 0.82 CYP3A4 (0.87) CYP3A4NAMPTXDHPARP1KDM4E
Ethyl Acetate SCHEMBL27415791 0.80 CYP3A4 (0.68) CYP3A4NAMPTXDHPARP1KDM4E
Alcohol SCHEMBL28252889 0.78 CYP3A4 (0.65) CYP3A4NAMPTXDHPARP1KDM4E
SCHEMBL29923659 0.77 CYP3A4 (0.77) CYP3A4NAMPTXDHPARP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110818710-B Benzodiazepine compound and preparation method thereof 石河子大学 2021-02-09 CN disclosed
CN-110818710-A Benzodiazepine compound and preparation method thereof 石河子大学 2020-02-21 CN disclosed