SCHEMBL28384265

SCHEMBL28384265

CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(C(=O)O)cc2)ncc1Cl

nearest known ligand 0.76

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 12/20 0.76
HDAC1 Q13547 3/20 0.76
PTK2 Q05397 7/20 0.70
HDAC2 Q92769 2/20 0.68
HDAC6 Q9UBN7 2/20 0.68
AURKA O14965 1/20 0.68
MET P08581 5/20 0.66
INSR P06213 1/20 0.63
ROS1 P08922 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11916626 0.91 ALK (0.77) ALKHDAC1PTK2HDAC2HDAC6
SCHEMBL28387246 0.86 ALK (1.00) ALKHDAC1PTK2HDAC2HDAC6
SCHEMBL18350626 0.86 ALK (0.83) ALKHDAC1METINSRROS1
SCHEMBL21437921 0.86 AXL (0.70) ALKHDAC1PTK2HDAC2HDAC6
SCHEMBL11901091 0.84 ALK (0.73) ALKHDAC1PTK2HDAC2HDAC6
SCHEMBL23534017 0.84 ALK (0.70) ALKHDAC1PTK2HDAC2HDAC6
SCHEMBL29805788 0.84 ALK (0.70) ALKHDAC1PTK2HDAC2HDAC6
SCHEMBL29805808 0.83 ALK (0.68) ALKHDAC1PTK2HDAC2HDAC6
SCHEMBL26716965 0.83 ALK (0.68) ALKHDAC1PTK2HDAC2HDAC6
SCHEMBL17481584 0.83 PTK2 (0.68) ALKHDAC1PTK2HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111039875-A HDAC/ALK double-target-point inhibitor and preparation method and application thereof 重庆医科大学 2020-04-21 CN disclosed