SCHEMBL28397182

SCHEMBL28397182

[CH2]c1ccc(-c2nnc(-c3nc(-c4ccc(S(=O)(=O)C(C)C)cc4F)cnc3N(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)o2)cc1

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ATR Q13535 19/20 0.44
GSK3B P49841 1/20 0.44
PRKDC P78527 1/20 0.44
FEN1 P39748 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2486124 0.89 ATR (0.42) ATRGSK3BPRKDC
SCHEMBL20420666 0.89 ATR (0.43) ATRGSK3BPRKDC
SCHEMBL16420825 0.80 ATR (0.50) ATRGSK3BPRKDC
SCHEMBL16491618 0.79 ATR (0.47) ATRGSK3BPRKDC
SCHEMBL2509496 0.79 ATR (0.48) ATRGSK3BPRKDC
SCHEMBL16489081 0.79 ATR (0.47) ATRGSK3BPRKDC
SCHEMBL2483790 0.77 ATR (0.51) ATRGSK3BPRKDC
SCHEMBL20738904 0.77 ATR (0.45) ATRGSK3BPRKDC
SCHEMBL16420823 0.76 ATR (0.49) ATRGSK3BPRKDC
SCHEMBL2482615 0.75 ATR (0.45) ATRGSK3BPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106496209-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2020-06-30 CN disclosed
CN-106496210-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2020-06-09 CN disclosed
CN-106518856-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2020-04-28 CN disclosed