SCHEMBL28398397

SCHEMBL28398397

C(=Cc1ccccn1)c1ccc(Nc2ccnc(NCc3ccccc3)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 2/20 0.49
MAPK8 P45983 1/20 0.49
MAPT P10636 4/20 0.48
AURKA O14965 2/20 0.48
PIM1 P11309 2/20 0.48
CHEK1 O14757 1/20 0.48
IKBKB O14920 1/20 0.48
NPC1 O15118 1/20 0.48
PDPK1 O15530 1/20 0.48
CHEK2 O96017 1/20 0.48
PRKCG P05129 1/20 0.48
CDK1 P06493 1/20 0.48
LYN P07948 1/20 0.48
KIT P10721 1/20 0.48
FGFR1 P11362 1/20 0.48
FGFR3 P22607 1/20 0.48
RPS6KB1 P23443 1/20 0.48
CDK2 P24941 1/20 0.48
MARK3 P27448 1/20 0.48
MAPK1 P28482 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29866713 1.00 CDC7 (0.49) CDC7MAPK8MAPTAURKAPIM1
SCHEMBL28395245 0.91 NPC1 (0.51) CDC7MAPK8MAPTAURKAPIM1
SCHEMBL29865902 0.91 NPC1 (0.51) CDC7MAPK8MAPTAURKAPIM1
SCHEMBL28396622 0.88 MAPT (0.54) MAPTNPC1FGFR1CDK2MAPK1
SCHEMBL29866340 0.87 AURKA (0.66) MAPK8MAPTAURKAPIM1CHEK1
SCHEMBL28398207 0.87 AURKA (0.66) MAPK8MAPTAURKAPIM1CHEK1
SCHEMBL28405713 0.81 AURKA (0.54) MAPTAURKAPIM1CHEK1IKBKB
SCHEMBL29866211 0.81 AURKA (0.54) MAPTAURKAPIM1CHEK1IKBKB
SCHEMBL28405661 0.79 AURKA (0.45) MAPK8MAPTAURKAPIM1CHEK1
SCHEMBL29866256 0.78 NPC1 (0.43) MAPTAURKAPIM1CHEK1IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111004215-B 2, 4-substituted pyrimidine derivatives, preparation method thereof and application thereof in preparing antitumor drugs 华北理工大学 2022-08-09 CN disclosed
CN-111004215-A 2, 4-substituted pyrimidine derivatives, preparation method thereof and application thereof in preparing antitumor drugs 华北理工大学 2020-04-14 CN disclosed