SCHEMBL28399032

SCHEMBL28399032

Nc1ncc(OC(=O)c2ccccc2)nc1C(=O)Nc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ATR Q13535 20/20 0.62
PRKDC P78527 6/20 0.60
ATM Q13315 2/20 0.56
CYP3A4 P08684 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL560180 0.82 ATR (0.65) ATRPRKDCATMCYP3A4
SCHEMBL559881 0.77 ATR (1.00) ATRPRKDCATMCYP3A4
SCHEMBL12186471 0.76 ATR (0.72) ATRPRKDCATMCYP3A4
SCHEMBL3860081 0.76 ATR (0.72) ATRPRKDCATMCYP3A4
SCHEMBL19152946 0.76 ATR (0.72) ATRPRKDCATMCYP3A4
SCHEMBL30667685 0.75 ATR (1.00) ATRPRKDCATMCYP3A4
SCHEMBL560845 0.75 ATR (0.70) ATRPRKDCATMCYP3A4
SCHEMBL2480842 0.75 ATR (1.00) ATRPRKDCATMCYP3A4
SCHEMBL2484673 0.73 ATR (1.00) ATRPRKDCATMCYP3A4
SCHEMBL30606835 0.72 ATR (1.00) ATRPRKDCATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106496209-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2020-06-30 CN disclosed
CN-106496210-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2020-06-09 CN disclosed
CN-106518856-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2020-04-28 CN disclosed