SCHEMBL28399652

SCHEMBL28399652

CN1CC(Br)=CC=C1C1=CCNCC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.46
SIGMAR1 Q99720 2/20 0.39
QDPR P09417 2/20 0.37
HTR6 P50406 2/20 0.35
HTR2A P28223 1/20 0.35
HTR7 P34969 1/20 0.35
LMNA P02545 1/20 0.34
BLM P54132 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
DRD2 P14416 1/20 0.34
ALOX15 P16050 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CDK9 P50750 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL25217174 0.64 HTR2C (1.00) HTR2CSIGMAR1QDPRHTR6HTR2A
SCHEMBL21246808 0.64 HTR2C (0.38) HTR2CSIGMAR1QDPRHTR6HTR2A
SCHEMBL24402613 0.62
SCHEMBL1199051 0.61 HTR2C (1.00) HTR2CSIGMAR1QDPRHTR6HTR2A
Hydrochloric Acid SCHEMBL28666550 0.61 HTR2C (0.47) HTR2CSIGMAR1QDPRHTR6HRH3
SCHEMBL4790160 0.61 HTR2C (0.61) HTR2CSIGMAR1QDPRHTR6HTR2A
Hydrochloric Acid SCHEMBL20292040 0.60 HTR2C (0.42) HTR2CSIGMAR1QDPRHTR6HTR2A
SCHEMBL28506378 0.60 HTR2C (0.60) HTR2CSIGMAR1QDPRHTR6HTR2A
SCHEMBL3666854 0.60 HTR2C (0.38) HTR2CSIGMAR1QDPRHTR6HTR2A
Hydrochloric Acid SCHEMBL7290341 0.60 HTR2C (0.67) HTR2CSIGMAR1QDPRHTR6HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115710266-A Pyridopyrimidine derivative, preparation method thereof and application thereof in medicines 江苏恒瑞医药股份有限公司 2023-02-24 CN disclosed
CN-111094289-B Pyridopyrimidine derivative, preparation method thereof and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed
CN-113082224-A Pyridopyrimidine derivative conjugate, preparation method thereof and application thereof in medicines 江苏恒瑞医药股份有限公司 2021-07-09 CN disclosed
CN-111094289-A Pyridopyrimidine derivative, preparation method thereof and application thereof in medicine 江苏恒瑞医药股份有限公司 2020-05-01 CN disclosed