SCHEMBL28401049

SCHEMBL28401049

CC(C)(C)OC(=O)N1C[C@@H](O)C[C@@H]1C(=O)Nc1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 3/20 0.60
BCR P11274 3/20 0.60
POLB P06746 3/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2C19 P33261 1/20 0.56
KMT2A Q03164 2/20 0.50
MAPT P10636 1/20 0.48
EPHX2 P34913 1/20 0.47
KDR P35968 1/20 0.46
RECQL P46063 1/20 0.44
GRIN2B Q13224 1/20 0.44
MEN1 O00255 1/20 0.44
PDK1 Q15118 1/20 0.43
TSHR P16473 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HDAC8 Q9BY41 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28395665 0.91 ABL1 (0.61) ABL1BCRPOLBCYP1A2CYP3A4
SCHEMBL28396799 0.87 ABL1 (0.55) ABL1BCRPOLBCYP1A2CYP3A4
SCHEMBL2568434 0.87 POLB (0.57) ABL1BCRPOLBCYP1A2CYP3A4
SCHEMBL31122514 0.86 POLB (0.58) ABL1BCRPOLBCYP1A2CYP3A4
SCHEMBL28993060 0.85 ABL1 (0.55) ABL1BCRPOLBCYP1A2CYP3A4
SCHEMBL28993059 0.85 ABL1 (0.55) ABL1BCRPOLBCYP1A2CYP3A4
SCHEMBL28392847 0.85 ABL1 (0.55) ABL1BCRPOLBCYP1A2CYP3A4
SCHEMBL28733147 0.85 ABL1 (0.55) ABL1BCRPOLBCYP1A2CYP3A4
SCHEMBL29639985 0.83 NPC1 (0.63) ABL1BCRCYP1A2CYP3A4CYP2C19
SCHEMBL7722205 0.80 NPC1 (0.62) POLBCYP1A2CYP3A4CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109761957-B Hydroxyproline-containing compound and preparation method and application thereof 西安交通大学 2020-05-19 CN claimed
CN-109796439-B Hydroxyproline peptide derivative and preparation method and application thereof 西安交通大学 2020-05-19 CN claimed
CN-109796439-B Hydroxyproline peptide derivative and preparation method and application thereof 西安交通大学 2020-05-19 CN disclosed
CN-109761957-B Hydroxyproline-containing compound and preparation method and application thereof 西安交通大学 2020-05-19 CN disclosed