SCHEMBL28401968

SCHEMBL28401968

Cc1nn(C2CCOCC2)c2cc(O)ccc12

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.49
PIK3CD O00329 2/20 0.47
SPR P35270 2/20 0.46
PDE7A Q13946 9/20 0.40
PDE1A P54750 2/20 0.39
PDE1B Q01064 2/20 0.39
PDE1C Q14123 2/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PDE4D Q08499 1/20 0.38
CFTR P13569 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19703379 0.86 PIK3CD (0.48) PIK3CDSPRPDE7APDE1APDE1B
SCHEMBL28410346 0.83 PIK3CD (0.47) PIK3CDSPRPDE7APDE1APDE1B
SCHEMBL30619300 0.83 PIK3CD (0.47) PIK3CDSPRPDE7APDE1APDE1B
SCHEMBL19698034 0.81 PIK3CD (0.46) PIK3CDSPRPDE7APDE1APDE1B
SCHEMBL28398423 0.76 PIK3CD (0.42) PIK3CDSPRPDE7APDE1APDE1B
SCHEMBL19597133 0.75 KDM4C (0.50) PIK3CDSPRPDE7APDE1APDE1B
SCHEMBL18731891 0.74 PIK3CD (0.38) ESR1PIK3CDPDE1APDE1BPDE1C
SCHEMBL28396902 0.73 PIK3CD (0.44) PIK3CDSPRPDE1APDE1BPDE1C
SCHEMBL30619306 0.73 PIK3CD (0.44) PIK3CDSPRPDE1APDE1BPDE1C
SCHEMBL18731899 0.72 ESR1 (0.42) ESR1PIK3CDPDE7AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111196804-B TGF-beta R1 inhibitors and uses thereof 南京圣和药业股份有限公司 2023-11-07 CN disclosed
CN-111196804-A TGF- β R1 inhibitor and application thereof 南京圣和药业股份有限公司 2020-05-26 CN disclosed