SCHEMBL28414296

SCHEMBL28414296

O=C1Nc2ccc([N+](=O)[O-])cc2C1=C(Nc1ccccc1)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.55
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
CAPN9 O14815 1/20 0.51
CASP3 P42574 1/20 0.51
TGM2 P21980 1/20 0.45
CXCR1 P25024 1/20 0.44
CXCR2 P25025 1/20 0.44
GSK3B P49841 3/20 0.44
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA9 Q16790 2/20 0.44
POLB P06746 2/20 0.44
NPC1 O15118 1/20 0.44
MITF O75030 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPT P10636 3/20 0.44
GAA P10253 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29642973 1.00 EGFR (0.55) EGFRMEN1KMT2ACAPN9CASP3
SCHEMBL6319460 0.97 EGFR (0.54) EGFRMEN1KMT2ACAPN9CASP3
SCHEMBL6319442 0.97 EGFR (0.54) EGFRMEN1KMT2ACAPN9CASP3
SCHEMBL8010041 0.93 EGFR (0.51) EGFRMEN1KMT2ACAPN9CASP3
SCHEMBL6320292 0.93 EGFR (0.51) EGFRMEN1KMT2ACAPN9CASP3
SCHEMBL6326010 0.92 EGFR (0.50) EGFRMEN1KMT2ACAPN9CASP3
SCHEMBL6326004 0.92 EGFR (0.50) EGFRMEN1KMT2ACAPN9CASP3
SCHEMBL6322554 0.92 EGFR (0.50) EGFRMEN1KMT2ACAPN9CASP3
SCHEMBL6322561 0.92 EGFR (0.50) EGFRMEN1KMT2ACAPN9CASP3
SCHEMBL6318752 0.92 EGFR (0.50) EGFRMEN1KMT2ACAPN9CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111285872-B Indole-2-ketone derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2022-05-17 CN disclosed
CN-111285872-A Indole-2-ketone derivative and preparation method and application thereof 北京志健金瑞生物医药科技有限公司 2020-06-16 CN disclosed