SCHEMBL28415482

SCHEMBL28415482

Cc1cc(C2CCC(C(C)NC(=NC#N)Nc3ccc(Cl)cc3)CC2)ccn1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 13/20 0.61
CYP2C9 P11712 3/20 0.37
CYP2C8 P10632 2/20 0.37
TDO2 P48775 2/20 0.37
CHRNA1 P02708 1/20 0.37
CYP2C19 P33261 1/20 0.37
CYP3A4 P08684 1/20 0.37
KCNH2 Q12809 1/20 0.37
PRCP P42785 1/20 0.35
KCNJ11 Q14654 1/20 0.33
MAPK1 P28482 2/20 0.33
USP30 Q70CQ3 1/20 0.33
TLR8 Q9NR97 1/20 0.32
TLR7 Q9NYK1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187200 1.00 IDO1 (0.61) IDO1CYP2C9CYP2C8TDO2CHRNA1
SCHEMBL21187212 0.88 IDO1 (0.64) IDO1CYP2C9CYP2C8TDO2CHRNA1
SCHEMBL21187192 0.82 IDO1 (0.68) IDO1CYP2C9CYP2C8TDO2CHRNA1
SCHEMBL28414622 0.78 IDO1 (0.73) IDO1CYP2C9CYP2C8TDO2CHRNA1
SCHEMBL23111225 0.76 IDO1 (1.00) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL17742848 0.76 IDO1 (1.00) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL17742849 0.76 IDO1 (1.00) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL18864223 0.76 IDO1 (1.00) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL17730125 0.76 IDO1 (1.00) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL20838627 0.76 IDO1 (0.64) IDO1CYP2C9CYP2C8TDO2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111247119-B Amidine and guanidine derivatives, preparation method and application thereof in medicines 四川科伦博泰生物医药股份有限公司 2023-02-03 CN disclosed
CN-111247119-A Amidine and guanidine derivatives, preparation method and application thereof in medicines 四川科伦博泰生物医药股份有限公司 2020-06-05 CN disclosed