SCHEMBL28419637

SCHEMBL28419637

Cc1c(-c2cccc(O)c2F)c(=O)n(CC(OC(N)=O)c2ccccc2)c(=O)n1Cc1c(F)cccc1C(F)(F)F

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 20/20 0.65
CYP3A4 P08684 14/20 0.65
ADRB2 P07550 1/20 0.57
APLNR P35414 1/20 0.57
OPRK1 P41145 1/20 0.57
GLP1R P43220 1/20 0.57
CX3CR1 P49238 1/20 0.57
FFAR4 Q5NUL3 1/20 0.57
GPR119 Q8TDV5 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20547876 0.92 GNRHR (0.78) GNRHRCYP3A4ADRB2APLNROPRK1
SCHEMBL20547877 0.92 GNRHR (0.78) GNRHRCYP3A4ADRB2APLNROPRK1
SCHEMBL28421982 0.90 GNRHR (0.67) GNRHRCYP3A4ADRB2APLNROPRK1
SCHEMBL28419485 0.88 GNRHR (0.79) GNRHRCYP3A4
SCHEMBL28419487 0.88 GNRHR (0.79) GNRHRCYP3A4
SCHEMBL28418291 0.87 GNRHR (0.62) GNRHRCYP3A4
SCHEMBL28418260 0.86 GNRHR (0.54) GNRHRCYP3A4
SCHEMBL28421910 0.85 GNRHR (0.61) GNRHRCYP3A4ADRB2APLNROPRK1
SCHEMBL28421914 0.84 GNRHR (0.59) GNRHRCYP3A4ADRB2APLNROPRK1
SCHEMBL28421940 0.84 GNRHR (0.59) GNRHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111333587-B Substituted pyrimidine-2, 4 (1H, 3H) -dione derivatives and uses thereof 东莞市东阳光新药研发有限公司 2023-04-07 CN disclosed
CN-111333587-A Substituted pyrimidine-2, 4(1H,3H) -dione derivatives and uses thereof 东莞市东阳光新药研发有限公司 2020-06-26 CN disclosed