SCHEMBL28426652

SCHEMBL28426652

Cc1cccc2c1NCCCN2c1ccc(NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.40
CREBBP Q92793 1/20 0.40
AVPR2 P30518 1/20 0.39
AVPR1A P37288 1/20 0.39
NR1I3 Q14994 3/20 0.38
DRD2 P14416 1/20 0.38
LIPE Q05469 1/20 0.38
NAMPT P43490 1/20 0.38
CD274 Q9NZQ7 1/20 0.37
CYP17A1 P05093 2/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPT P10636 3/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 1/20 0.36
ACHE P22303 1/20 0.36
BACE1 P56817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16239010 0.73 P2RX4 (0.49) BRD4CREBBPNR1I3DRD2LIPE
SCHEMBL14525364 0.71 SMN1; SMN2 (0.53) DRD2ALDH1A1MAPTNPC1RAB9A
SCHEMBL6503210 0.69 MAPT (0.50) NAMPTCD274ALDH1A1MAPTKDM4E
SCHEMBL13055402 0.67 CYP17A1 (0.59) DRD2LIPENAMPTCYP17A1ALDH1A1
SCHEMBL27292734 0.67 NAMPT (0.49) DRD2LIPENAMPTALDH1A1MAPT
SCHEMBL1968536 0.66 DDB1 (0.45) BRD4CREBBPNR1I3NAMPTCYP17A1
SCHEMBL8346062 0.65 PRKDC (0.63) CD274ALDH1A1MAPTKDM4ENPC1
SCHEMBL993933 0.65 GAA (0.64) DRD2NAMPTMAPTNPC1RAB9A
SCHEMBL8739188 0.65 MAPT (0.58) ALDH1A1MAPTKDM4ENPC1RAB9A
SCHEMBL28392058 0.65 BRD4 (0.45) BRD4NAMPTCYP17A1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108863959-B P2X4 receptor antagonists 日本化学药品株式会社 2021-11-30 CN disclosed
CN-111333588-A P2X4 receptor antagonists 日本化学药品株式会社 2020-06-26 CN disclosed