Bromide

Bromide

SCHEMBL2842856

Br.CCCCc1nc(C)n(CCc2ccccc2)c(=O)c1Cc1ccc(-c2ccccc2-c2noc(=O)[nH]2)cc1

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPARG P37231 13/20 0.60
SLC33A1 O00400 2/20 0.55
AGTR1 P30556 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1891379 0.99 PPARG (0.61) PPARGSLC33A1AGTR1
Bromide SCHEMBL1889445 0.94 PPARG (0.59) PPARGSLC33A1AGTR1
SCHEMBL1889929 0.94 PPARG (0.63) PPARGSLC33A1AGTR1
Bromide SCHEMBL3565943 0.94 PPARG (0.58) PPARGSLC33A1AGTR1
SCHEMBL1891644 0.93 PPARG (0.59) PPARGSLC33A1AGTR1
Bromide SCHEMBL1890455 0.93 PPARG (0.54) PPARGSLC33A1AGTR1
Bromide SCHEMBL1895257 0.93 PPARG (0.68) PPARGAGTR1
SCHEMBL1894785 0.93 PPARG (0.59) PPARGSLC33A1AGTR1
Hydrochloric Acid SCHEMBL1896020 0.93 PPARG (0.59) PPARGSLC33A1AGTR1
SCHEMBL1896115 0.93 PPARG (0.59) PPARGSLC33A1AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2256115-A1 Heteromonocyclic compound and use thereof Takeda Pharmaceutical Company Limited (JP) 2010-12-01 EP disclosed