SCHEMBL28432121

SCHEMBL28432121

CC(C)OS(=O)(=O)CNC(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
CA12 O43570 7/20 0.41
CA1 P00915 6/20 0.41
CA14 Q9ULX7 4/20 0.41
CA7 P43166 3/20 0.41
TDP1 Q9NUW8 1/20 0.41
CA2 P00918 5/20 0.40
CTSS P25774 3/20 0.38
CTSK P43235 3/20 0.38
CA9 Q16790 3/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CYP2D6 P10635 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
MALT1 Q9UDY8 1/20 0.36
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28520649 0.85 CA12 (0.42) MEN1GAAKMT2ACA12CA1
SCHEMBL16100172 0.79 MEN1 (0.45) MEN1GAAKMT2ACA12CA1
SCHEMBL3458070 0.77 TDP1 (0.42) MEN1GAAKMT2ACA12CA1
SCHEMBL3809117 0.75 TDP1 (0.44) MEN1GAAKMT2ACA12CA1
SCHEMBL18343870 0.75 CA12 (0.44) MEN1GAAKMT2ACA12CA1
SCHEMBL30738873 0.74 TDP1 (0.46) MEN1GAAKMT2ACA12CA1
SCHEMBL569003 0.72 SERPINE1 (0.43) MEN1GAAKMT2ACA12CA1
SCHEMBL221274 0.71 KMT2A (0.41) MEN1GAAKMT2ACA12CA1
SCHEMBL3579459 0.71 KMT2A (0.41) MEN1GAAKMT2ACA12CA1
SCHEMBL4818756 0.71 KMT2A (0.41) MEN1GAAKMT2ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106714844-B Anthracycline disulfide intermediates, antibody-drug conjugates and methods 基因泰克公司 2022-08-05 CN disclosed
CN-107735399-B Chiral diaryl macrocycles as modulators of protein kinases 特普医药公司 2021-01-26 CN disclosed
CN-111971287-A Macrocyclic compounds as TRK kinase inhibitors 重庆复创医药研究有限公司 2020-11-20 CN disclosed
CN-106565696-B Oxadiazole derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2020-07-28 CN disclosed