SCHEMBL28435744

SCHEMBL28435744

O=C(OCc1ccccc1)N1CCN(C2CCCC2)C(=O)C1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.54
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
TMEM97 Q5BJF2 6/20 0.53
SIGMAR1 Q99720 6/20 0.53
HTR1A P08908 2/20 0.53
HRH2 P25021 2/20 0.53
HRH1 P35367 2/20 0.53
HRH3 Q9Y5N1 2/20 0.53
ADRA2C P18825 1/20 0.53
CHRM4 P08173 1/20 0.53
CHRM5 P08912 1/20 0.53
ADRA2A P08913 1/20 0.53
ADRA2B P18089 1/20 0.53
ADRA1D P25100 1/20 0.53
HTR2A P28223 1/20 0.53
HTR2C P28335 1/20 0.53
ADRA1A P35348 1/20 0.53
ADRA1B P35368 1/20 0.53
DRD3 P35462 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31461542 0.95 SMN1; SMN2 (0.56) SMN1; SMN2NPC1RAB9ATMEM97SIGMAR1
SCHEMBL3069766 0.90 SMN1; SMN2 (0.54) SMN1; SMN2NPC1RAB9ATMEM97SIGMAR1
SCHEMBL14334656 0.88 SMN1; SMN2 (0.58) SMN1; SMN2NPC1RAB9ATMEM97SIGMAR1
SCHEMBL21041191 0.88 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9ATMEM97SIGMAR1
SCHEMBL30283170 0.87 HTR2C (0.52) SMN1; SMN2NPC1RAB9ATMEM97SIGMAR1
SCHEMBL27242728 0.85 MEN1 (0.53) SMN1; SMN2NPC1RAB9ATMEM97SIGMAR1
SCHEMBL3069899 0.85 SMN1; SMN2 (0.49) SMN1; SMN2NPC1RAB9ATMEM97SIGMAR1
SCHEMBL30368837 0.85 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL12526593 0.85 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL21209423 0.83 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9ATMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107098886-B Prazinone-containing quinazolinone PARP-1/2 inhibitor and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2020-07-14 CN disclosed