SCHEMBL28436719

SCHEMBL28436719

Cc1cc(-c2ccc(O)c(C)c2)c2ccccc2n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.53
TLR8 Q9NR97 4/20 0.49
ALDH1A1 P00352 2/20 0.48
MAPT P10636 2/20 0.48
HPGD P15428 2/20 0.48
KDM4E B2RXH2 1/20 0.48
USP2 O75604 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
NCF1 P14598 1/20 0.46
HSD17B1 P14061 2/20 0.45
HSD17B2 P37059 2/20 0.45
AURKA O14965 1/20 0.45
AURKB Q96GD4 1/20 0.45
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43
TUBB4B P68371 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23496945 0.85 BACE1 (0.55) CYP1A2TLR8NCF1HSD17B1HSD17B2
SCHEMBL23496931 0.84 CYP1A2 (0.56) CYP1A2ALDH1A1MAPTHPGDKDM4E
SCHEMBL30719607 0.84 CYP1A2 (0.56) CYP1A2ALDH1A1MAPTHPGDKDM4E
SCHEMBL23496929 0.83 TLR8 (0.50) CYP1A2TLR8ALDH1A1MAPTKDM4E
SCHEMBL28129147 0.83 CYP1A2 (0.53) CYP1A2ALDH1A1MAPTHPGDKDM4E
SCHEMBL23496944 0.82 NT5E (0.49) CYP1A2TLR8HSD17B1HSD17B2CDC7
SCHEMBL30719595 0.82 NT5E (0.49) CYP1A2TLR8HSD17B1HSD17B2CDC7
SCHEMBL12834414 0.82 ERN1 (0.52) CYP1A2ALDH1A1MAPTHPGDKDM4E
SCHEMBL18731749 0.80 CYP1A2 (0.58) CYP1A2ALDH1A1MAPTHPGDKDM4E
SCHEMBL1104820 0.80 CYP1A2 (0.62) CYP1A2ALDH1A1MAPTHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117586108-A TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2024-02-23 CN claimed
CN-117659025-A TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2024-03-08 CN disclosed
CN-117586191-A TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2024-02-23 CN disclosed
CN-117586108-A TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2024-02-23 CN disclosed
CN-111542515-B TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2023-12-05 CN disclosed
CN-111542515-A TOLL-like receptor 8(TLR8) specific antagonist and preparation method and application thereof 科罗拉多州立大学董事会法人团体 2020-08-14 CN disclosed