SCHEMBL28449337

SCHEMBL28449337

CC(C)(OC(N)=O)C(=O)Nc1cc(Br)sc1C(N)=O

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 12/20 0.38
IRAK4 Q9NWZ3 1/20 0.32
CFTR P13569 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 1/20 0.32
RXFP1 Q9HBX9 1/20 0.30
RAF1 P04049 1/20 0.30
MAPK14 Q16539 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28453670 0.83 IKBKB (0.36) IKBKBRAF1MAPK14
SCHEMBL3610995 0.81 LCK (0.41) IKBKBRXFP1
SCHEMBL14343926 0.78 IKBKB (0.39) IKBKBIRAK4RXFP1
SCHEMBL6192110 0.76 LCK (0.38) IKBKBRXFP1
SCHEMBL490588 0.76 IKBKB (0.57) IKBKB
SCHEMBL20572261 0.75 IKBKB (0.47) IKBKBKDM4E
SCHEMBL28453667 0.73 IKBKB (0.34) IKBKBIRAK4
SCHEMBL28453668 0.73 IKBKB (0.34) IKBKBIRAK4
SCHEMBL28449106 0.73 IKBKB (0.38) IKBKBALDH1A1
SCHEMBL28449109 0.73 IKBKB (0.38) IKBKBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409373-A Substituted [5,6] cyclo-4 (3H) -pyrimidinones as anticancer agents 南京正济医药研究有限公司 2021-02-26 CN disclosed
CN-110381950-B Substituted [5,6] cyclo-4 (3H) -pyrimidinones as anticancer agents 南京正济医药研究有限公司 2020-09-04 CN disclosed