SCHEMBL28452907

SCHEMBL28452907

Clc1cccc(Nc2nc(OC3CCNCC3)c3cc[nH]c3n2)c1

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PAK4 O96013 6/20 0.67
CCNB2 O95067 1/20 0.44
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
CCNA2 P20248 1/20 0.44
CDK2 P24941 1/20 0.44
CCNA1 P78396 1/20 0.44
CCNB3 Q8WWL7 1/20 0.44
EGFR P00533 3/20 0.44
PDPK1 O15530 1/20 0.43
TTBK1 Q5TCY1 1/20 0.43
TTBK2 Q6IQ55 1/20 0.43
SYK P43405 1/20 0.43
TTK P33981 4/20 0.42
JAK2 O60674 1/20 0.41
BRD4 O60885 1/20 0.41
JAK3 P52333 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4920465 0.75 TTK (0.51) CDK1CCNB1CDK2EGFRPDPK1
SCHEMBL20654492 0.72 FLT3 (0.45) PAK4CCNB2CDK1CCNB1CCNA2
SCHEMBL23690869 0.69 JAK3 (0.62) EGFRJAK2JAK3
SCHEMBL31085501 0.69 JAK3 (0.62) EGFRJAK2JAK3
SCHEMBL28446369 0.68 PAK4 (1.00) PAK4TTBK1TTBK2
SCHEMBL28446370 0.68 PAK4 (1.00) PAK4TTBK1TTBK2
SCHEMBL28450012 0.68 PAK4 (1.00) PAK4TTBK1TTBK2
SCHEMBL20183342 0.67 JAK3 (0.76) JAK2JAK3
SCHEMBL28455827 0.66 PAK4 (0.78) PAK4
SCHEMBL28456610 0.65 PAK4 (0.65) PAK4TTBK1TTBK2TTKJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111620878-A Pyrrolopyrimidine derivatives as protein kinase inhibitors and application thereof 中国药科大学 2020-09-04 CN disclosed