SCHEMBL28455243

SCHEMBL28455243

OC1CCN(c2nc(Nc3ccc(C(F)(F)F)cc3)nc(Nc3cccc(C(F)(F)F)c3)n2)C1

nearest known ligand 0.92

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
IDH2 P48735 18/20 0.92
MAPT P10636 1/20 0.60
APP P05067 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30568848 0.96 IDH2 (1.00) IDH2MAPTAPP
SCHEMBL28450644 0.96 IDH2 (1.00) IDH2MAPTAPP
SCHEMBL28460705 0.96 IDH2 (1.00) IDH2MAPTAPP
SCHEMBL28450649 0.96 IDH2 (1.00) IDH2MAPTAPP
SCHEMBL30568844 0.96 IDH2 (1.00) IDH2MAPTAPP
SCHEMBL30568821 0.96 IDH2 (1.00) IDH2MAPTAPP
SCHEMBL28455232 0.91 IDH2 (0.90) IDH2MAPTAPP
SCHEMBL30568831 0.91 IDH2 (0.90) IDH2MAPTAPP
SCHEMBL28451068 0.90 IDH2 (0.88) IDH2MAPTAPP
SCHEMBL28456888 0.90 IDH2 (0.88) IDH2MAPTAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662242-B Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2023-10-24 CN disclosed
CN-111662242-A Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2020-09-15 CN disclosed