Atorvastatin

Atorvastatin

SCHEMBL28457

CC(C)c1c(C(=O)Nc2ccccc2)c(-c2ccccc2)c(-c2ccc(F)cc2)n1CC[C@@H](O)C[C@@H](O)CC(=O)O.[CaH2]

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HMGCR

The experimentally established mechanism targets of Atorvastatin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HMGCR known ✓ P04035 10/20 0.98
SLCO1B1 Q9Y6L6 4/20 0.98
ABCB11 O95342 3/20 0.98
HDAC1 Q13547 2/20 0.98
HDAC2 Q92769 2/20 0.98
HDAC6 Q9UBN7 2/20 0.98
NR1I2 O75469 1/20 0.98
RHOC P08134 1/20 0.98
CYP3A4 P08684 1/20 0.98
THRB P10828 1/20 0.98
NR1H4 Q96RI1 1/20 0.98
ABCG2 Q9UNQ0 1/20 0.98
ABCC3 O15438 2/20 0.86
ABCC4 O15439 2/20 0.86
SLCO1B3 Q9NPD5 2/20 0.86
PDE6D O43924 3/20 0.76
ABCB1 P08183 1/20 0.57
ABCC2 Q92887 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Atorvastatin SCHEMBL7037657 1.00 HMGCR (0.98) HMGCRSLCO1B1ABCB11HDAC1HDAC2
Atorvastatin SCHEMBL4994180 1.00 HMGCR (0.98) HMGCRSLCO1B1ABCB11HDAC1HDAC2
Atorvastatin SCHEMBL28270206 1.00 HMGCR (0.98) HMGCRSLCO1B1ABCB11HDAC1HDAC2
Atorvastatin SCHEMBL28252417 0.99 HMGCR (0.97) HMGCRSLCO1B1ABCB11HDAC1HDAC2
Atorvastatin SCHEMBL19469652 0.99 HMGCR (0.97) HMGCRSLCO1B1ABCB11HDAC1HDAC2
SCHEMBL6761283 0.99 HMGCR (0.97) HMGCRSLCO1B1ABCB11HDAC1HDAC2
Atorvastatin SCHEMBL26978250 0.99 HMGCR (0.97) HMGCRSLCO1B1ABCB11HDAC1HDAC2
Atorvastatin SCHEMBL34266 0.99 HMGCR (0.97) HMGCRSLCO1B1ABCB11HDAC1HDAC2
Atorvastatin SCHEMBL5799062 0.99 HMGCR (0.97) HMGCRSLCO1B1ABCB11HDAC1HDAC2
Atorvastatin SCHEMBL14968747 0.99 HMGCR (0.97) HMGCRSLCO1B1ABCB11HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 16450 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS CENTRE FOR DIGESTIVE DISEASES (AU) 2026-05-21 US claimed
EP-3982211-B1 METHOD AND DEVICE FOR SIMULATING PROCESSING ON A MACHINE TOOL BY MEANS OF A SELF-LEARNING SYSTEM DMG MORI DIGITAL GMBH (DE) 2026-05-13 EP claimed
EP-3545882-B1 APPARATUS TO ACCOUNT FOR TRANSPONDER TAGGED OBJECTS USED DURING CLINICAL PROCEDURES, EMPLOYING A TROCAR COVIDIEN LP (US) 2026-05-06 EP claimed
EP-4515141-B1 LIGHTING DEVICE WITH BENT LIGHT GUIDE(S) STELLANTIS AUTO SAS (FR) 2026-04-29 EP claimed
EP-3498548-B2 LIFTING SUPPORT ASSEMBLY WITH A SECURING DEVICE KOBER GMBH A (DE) 2026-04-29 EP claimed
EP-4446870-B1 TENSOR CALCULATION UNIT AND USE METHOD, AND DATA PROCESSING APPARATUS AND OPERATION METHOD HYGON INFORMATION TECHNOLOGY CO LTD (CN) 2026-04-29 EP claimed
EP-4092718-B1 LIQUID CHEMICAL PROCESSING DEVICE DAIKIN FINETECH LTD (JP) 2026-04-22 EP claimed
EP-4428800-B1 FRAUD DETECTION SYSTEM AT GAME PARLOR ANGEL PLAYING CARDS CO LTD (JP) 2026-04-22 EP claimed
EP-3839694-B1 PHOTOELECTRIC COMPUTING UNIT, PHOTOELECTRIC COMPUTING ARRAY, AND PHOTOELECTRIC COMPUTING METHOD NANJING UNIVERSITY (CN) 2026-04-15 EP claimed
EP-3955431-B1 STATOR ASSEMBLY, ELECTRIC MOTOR, COMPRESSOR, AND REFRIGERATION DEVICE ANHUI MEIZHI PREC MANUFACTURING CO LTD (CN) 2026-03-25 EP claimed
EP-0021853-B1 SELF-SCANNED ARRAYS OF PHOTOSENSORS XEROX CORPORATION (US) 1983-11-09 EP claimed
EP-0005267-B1 DEVICE FOR GLUEING PROTECTION POCKETS ONTO ALBUM SHEETS Heinz Beck, Kunststoffverarbeitung GmbH (DE) 1983-02-16 EP claimed
EP-0012196-B1 DEVICE FOR TRANSFERRING A STACK OF PRINTED MATTER FROM THE POSTS OF A FILING BINDER OR THE LIKE ONTO A BUNDLING MEMBER Willi G. Sonntag GmbH (DE) 1983-01-26 EP claimed
EP-0052174-A1 Filter press Parmentier, Alfred Henri (BE) 1982-05-26 EP claimed
EP-0051001-A1 Detergent container with a telescopic funnel, and laundry washing machine with at least one such container ESSWEIN S.A. (FR) 1982-05-05 EP claimed
EP-0002031-B1 METHODS OF INHIBITING PLANT AND COMBATING WEEDS USING ALPHA-AMINOALKANEPHOSPHONOUS ACIDS CIBA-GEIGY AG (CH) 1982-02-03 EP claimed
EP-0027802-A1 MOTOR VEHICLE FOR COMBINED TRANSPORT SYSTEMS BUNOUST, Christine (MC) 1981-05-06 EP claimed
WO-1980002265-A1 MOTOR VEHICLE FOR COMBINED TRANSPORT SYSTEMS BUNOUST C (MC) 1980-10-30 WO claimed
EP-0004340-B1 PSEUDORANDOM GENERATION OF ORTHOGONAL MATRIXES FOR SCRAMBLING PURPOSES Felten & Guilleaume Fernmeldeanlagen GmbH (DE) 1980-10-15 EP claimed
EP-0010491-A1 Support for a computer terminal Compagnie du RONEO société anonyme (FR) 1980-04-30 EP claimed