SCHEMBL28457628

SCHEMBL28457628

COc1ccc2c(c1)CCN(c1ccccc1)C2

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 10/20 0.62
DRD5 P21918 9/20 0.62
DRD2 P14416 8/20 0.56
DRD3 P35462 8/20 0.56
DRD4 P21917 6/20 0.56
AOC3 Q16853 1/20 0.55
MAOB P27338 1/20 0.50
LMNA P02545 1/20 0.50
MAPT P10636 1/20 0.50
ESR1 P03372 1/20 0.49
ESR2 Q92731 1/20 0.49
HRH1 P35367 1/20 0.48
HRH3 Q9Y5N1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5525452 0.91 DRD1 (0.57) DRD1DRD5DRD2DRD3DRD4
SCHEMBL10673137 0.85 DRD1 (0.52) DRD1DRD5DRD2DRD3DRD4
SCHEMBL29500325 0.85 MAOB (0.70) DRD1DRD5DRD2DRD3DRD4
SCHEMBL16827433 0.85 MAOB (0.70) DRD1DRD5DRD2DRD3DRD4
SCHEMBL29500341 0.85 EED (0.59) DRD1DRD5DRD2DRD3DRD4
SCHEMBL29500309 0.85 DRD1 (0.52) DRD1DRD5DRD2DRD3DRD4
SCHEMBL2948505 0.84 AKR1C3 (0.56) DRD1DRD5DRD2DRD3MAOB
SCHEMBL29500368 0.84 DRD1 (0.51) DRD1DRD5DRD2DRD3DRD4
SCHEMBL30296979 0.83 DRD1 (0.56) DRD1DRD5DRD2DRD3DRD4
SCHEMBL27806895 0.83 DRD1 (0.56) DRD1DRD5DRD2DRD3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111285804-B Method for synthesizing thioamide compound 广州中医药大学(广州中医药研究院) 2022-01-07 CN claimed
CN-111285804-A Method for synthesizing thioamide compound 广州中医药大学(广州中医药研究院) 2020-06-16 CN claimed
CN-111285804-B Method for synthesizing thioamide compound 广州中医药大学(广州中医药研究院) 2022-01-07 CN disclosed
CN-111285804-A Method for synthesizing thioamide compound 广州中医药大学(广州中医药研究院) 2020-06-16 CN disclosed