SCHEMBL28459472

SCHEMBL28459472

Nc1nc(Nc2cccc(C(F)(F)F)c2)nc(N2CCCC(N)C2)n1

nearest known ligand 0.90

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDH2 P48735 15/20 0.90
MAPT P10636 2/20 0.65
CAMK1D Q8IU85 3/20 0.61
MAP3K7 O43318 1/20 0.61
CSF1R P07333 1/20 0.61
PIM1 P11309 1/20 0.61
MAPK3 P27361 1/20 0.61
MAPK1 P28482 1/20 0.61
SYK P43405 1/20 0.61
BLK P51451 1/20 0.61
RIPK4 P57078 1/20 0.61
CSNK2A1 P68400 1/20 0.61
KCNH2 Q12809 1/20 0.61
MAP2K5 Q13163 1/20 0.61
MAP3K11 Q16584 1/20 0.61
AURKB Q96GD4 1/20 0.61
LMNA P02545 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30568819 0.95 IDH2 (1.00) IDH2MAPTCAMK1DMAP3K7CSF1R
SCHEMBL28456851 0.87 IDH2 (0.89) IDH2MAPTLMNA
SCHEMBL28450626 0.86 IDH2 (0.86) IDH2MAPTLMNA
SCHEMBL28451697 0.82 IDH2 (1.00) IDH2MAPT
SCHEMBL30568829 0.82 IDH2 (1.00) IDH2MAPT
SCHEMBL28460673 0.82 IDH2 (1.00) IDH2MAPT
SCHEMBL30568801 0.82 IDH2 (1.00) IDH2MAPT
SCHEMBL28451696 0.82 IDH2 (1.00) IDH2MAPT
SCHEMBL30568818 0.82 IDH2 (1.00) IDH2MAPT
SCHEMBL30568805 0.82 IDH2 (1.00) IDH2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662242-B Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2023-10-24 CN disclosed
CN-111662242-A Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2020-09-15 CN disclosed