SCHEMBL28463572

SCHEMBL28463572

O=C(NCCO)C(Cc1ccc(O)c(Br)c1)=NO

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 13/20 0.77
HDAC6 Q9UBN7 10/20 0.77
CA12 O43570 4/20 0.73
CA1 P00915 4/20 0.73
CA2 P00918 4/20 0.73
CA9 Q16790 4/20 0.73
CA4 P22748 1/20 0.73
CA6 P23280 1/20 0.73
CA5A P35218 1/20 0.73
CA7 P43166 1/20 0.73
CA13 Q8N1Q1 1/20 0.73
CA14 Q9ULX7 1/20 0.73
HDAC3 O15379 8/20 0.70
HDAC2 Q92769 6/20 0.70
NCOR2 Q9Y618 4/20 0.70
HDAC7 Q8WUI4 5/20 0.70
HDAC8 Q9BY41 5/20 0.70
HDAC4 P56524 4/20 0.70
HDAC10 Q969S8 4/20 0.70
HDAC11 Q96DB2 4/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29940238 1.00 HDAC1 (0.77) HDAC1HDAC6CA12CA1CA2
SCHEMBL28463571 1.00 HDAC1 (0.77) HDAC1HDAC6CA12CA1CA2
Hemibastadin 1 SCHEMBL4751505 0.89 PLK4 (0.82) HDAC1HDAC6CA12CA1CA2
SCHEMBL28449765 0.88 HDAC1 (0.75) HDAC1HDAC6CA12CA1CA2
SCHEMBL28449763 0.88 HDAC1 (0.75) HDAC1HDAC6CA12CA1CA2
SCHEMBL29939752 0.88 HDAC1 (0.75) HDAC1HDAC6CA12CA1CA2
SCHEMBL22401371 0.87 HDAC1 (1.00) HDAC1HDAC6CA12CA1CA2
Psammaplin A SCHEMBL12521616 0.87 HDAC1 (0.91) HDAC1HDAC6CA12CA1CA2
Psammaplin A SCHEMBL29367050 0.87 HDAC1 (0.91) HDAC1HDAC6CA12CA1CA2
Psammaplin A SCHEMBL364511 0.87 HDAC1 (0.91) HDAC1HDAC6CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111548286-A PSA derivative with HDAC3 inhibitory activity and application thereof 沈阳药科大学 2020-08-18 CN claimed
CN-111548286-B PSA derivative with HDAC3 inhibitory activity and application thereof 沈阳药科大学 2022-09-06 CN disclosed
CN-111548286-A PSA derivative with HDAC3 inhibitory activity and application thereof 沈阳药科大学 2020-08-18 CN disclosed