SCHEMBL28468898

SCHEMBL28468898

C=C/C=C/C(=O)Nc1cc(Nc2nccc(-c3cnn4ccccc34)n2)c(OC)cc1N1CC(N(C)C)C1

nearest known ligand 0.70

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.70
IGF1R P08069 3/20 0.69
KCNH2 Q12809 3/20 0.69
INSR P06213 2/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28942095 1.00 EGFR (0.70) EGFRIGF1RKCNH2INSR
SCHEMBL28471883 0.95 EGFR (0.70) EGFRIGF1RKCNH2INSR
SCHEMBL28942033 0.95 EGFR (0.70) EGFRIGF1RKCNH2INSR
SCHEMBL14719238 0.93 EGFR (0.80) EGFRIGF1RKCNH2INSR
SCHEMBL28963872 0.90 EGFR (0.87) EGFRIGF1RKCNH2
SCHEMBL28463739 0.90 EGFR (0.87) EGFRIGF1RKCNH2
SCHEMBL28469668 0.89 EGFR (0.88) EGFRIGF1RKCNH2INSR
SCHEMBL28942072 0.89 EGFR (0.88) EGFRIGF1RKCNH2INSR
SCHEMBL14719111 0.88 EGFR (0.79) EGFRIGF1RKCNH2INSR
SCHEMBL28942081 0.87 EGFR (0.73) EGFRIGF1RKCNH2INSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108191861-B N- [5- (pyrimidin-2-amino) -2, 4-disubstituted-phenyl ] -trans-2, 4-pentadiene-amide 天津大学 2020-10-02 CN disclosed