SCHEMBL28475196

SCHEMBL28475196

Fc1cc(C(F)(F)F)ccc1C=Cc1nc(COc2ccc(CCCCn3cncn3)cc2)co1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 4/20 0.59
MINK1 Q8N4C8 1/20 0.59
ALDH1A1 P00352 3/20 0.40
ALOX15 P16050 2/20 0.38
KDM4E B2RXH2 2/20 0.38
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
TP53 P04637 2/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
MAPK1 P28482 1/20 0.36
HMOX1 P09601 1/20 0.35
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22397959 1.00 ERBB2 (0.59) ERBB2MINK1ALDH1A1ALOX15KDM4E
SCHEMBL22397920 0.91 ERBB2 (0.57) ERBB2MINK1ALDH1A1ALOX15KDM4E
SCHEMBL28476961 0.91 ERBB2 (0.57) ERBB2MINK1ALDH1A1ALOX15KDM4E
SCHEMBL22397990 0.89 ERBB2 (0.63) ERBB2MINK1MAPTHMOX1
SCHEMBL22398092 0.89 ERBB2 (0.63) ERBB2MINK1MAPTHMOX1
SCHEMBL22398026 0.89 ERBB2 (0.60) ERBB2MINK1HMOX1
SCHEMBL22398024 0.89 ERBB2 (0.60) ERBB2MINK1HMOX1
SCHEMBL22397918 0.88 ERBB2 (0.62) ERBB2MINK1HMOX1
SCHEMBL22397921 0.88 ERBB2 (0.62) ERBB2MINK1HMOX1
SCHEMBL22398004 0.88 ERBB2 (0.57) ERBB2MINK1HMOX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111886234-B Heterocyclic mitochondrial activity inhibitors and uses thereof 蒙特利尔大学 2023-12-15 CN disclosed
CN-111886234-A Heterocyclic mitochondrial activity inhibitors and uses thereof 蒙特利尔大学 2020-11-03 CN disclosed