SCHEMBL28475211

SCHEMBL28475211

Fc1ccc(Nc2ncnc3ccc(I)cc23)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD38 P28907 1/20 0.62
LMNA P02545 5/20 0.60
CYP1A2 P05177 4/20 0.60
CYP3A4 P08684 4/20 0.60
CYP2D6 P10635 4/20 0.60
CYP2C19 P33261 4/20 0.60
USP2 O75604 3/20 0.60
CLK4 Q9HAZ1 3/20 0.60
HIF1A Q16665 3/20 0.60
MEN1 O00255 3/20 0.60
KMT2A Q03164 3/20 0.60
TSHR P16473 2/20 0.60
ALDH1A1 P00352 2/20 0.60
EGFR P00533 6/20 0.59
RAF1 P04049 1/20 0.55
BRAF P15056 1/20 0.55
TP53 P04637 1/20 0.55
MAPT P10636 2/20 0.53
HPGD P15428 1/20 0.53
MAPK1 P28482 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27878333 0.88 USP2 (0.65) CD38LMNACYP1A2CYP3A4CYP2D6
SCHEMBL28469603 0.85 MAPK1 (0.65) CD38LMNAMEN1KMT2AALDH1A1
SCHEMBL28471823 0.85 KDM4E (0.72) CD38LMNACYP1A2CYP3A4CYP2D6
SCHEMBL3007586 0.85 ALK (0.72) LMNAMEN1KMT2AALDH1A1EGFR
SCHEMBL15587953 0.85 CD38 (0.64) CD38LMNACYP1A2CYP3A4CLK4
SCHEMBL29971755 0.85 EGFR (0.70) CD38LMNACYP1A2CYP3A4CYP2D6
SCHEMBL1192879 0.85 EGFR (0.70) CD38LMNACYP1A2CYP3A4CYP2D6
SCHEMBL5740246 0.85 CNR1 (0.62) CD38LMNAMEN1KMT2ATSHR
SCHEMBL29058751 0.85 EGFR (0.71) CD38EGFRRAF1BRAFMAPK1
SCHEMBL30395473 0.85 EGFR (0.71) CD38EGFRRAF1BRAFMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107652275-B Quinazoline derivative and preparation method and application thereof 沈阳工业大学 2020-09-22 CN disclosed