SCHEMBL28477476

SCHEMBL28477476

COc1ccc(-c2ccc3nc([Se]CC(OC)OC)ccc3c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
PDGFRB P09619 2/20 0.40
PDGFRA P16234 2/20 0.40
CYP17A1 P05093 2/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
RECQL P46063 1/20 0.38
NCF1 P14598 1/20 0.38
HSD17B1 P14061 1/20 0.38
HSD17B2 P37059 1/20 0.38
CYP11B1 P15538 4/20 0.37
CYP11B2 P19099 4/20 0.37
NPC1 O15118 1/20 0.37
NFKB1 P19838 1/20 0.37
RAB9A P51151 1/20 0.37
NFKB2 Q00653 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29935562 1.00 HDAC2 (0.42) HDAC2HDAC8HDAC6PDGFRBPDGFRA
SCHEMBL22534287 0.79 BACE1 (0.41) HDAC2PDGFRBPDGFRAPOLBMAPT
SCHEMBL29935347 0.79 BACE1 (0.41) HDAC2PDGFRBPDGFRAPOLBMAPT
SCHEMBL29935519 0.75 HDAC2 (0.43) HDAC2HDAC8HDAC6PDGFRBPDGFRA
SCHEMBL22534298 0.75 HDAC2 (0.43) HDAC2HDAC8HDAC6PDGFRBPDGFRA
SCHEMBL29935360 0.75 NQO1 (0.40) NQO1
SCHEMBL22534227 0.75 CYP1A2 (0.39) KDM4EALDH1A1NCF1NPC1NFKB1
SCHEMBL22534224 0.74 HDAC2 (0.42) HDAC2HDAC8HDAC6PDGFRBPDGFRA
SCHEMBL29935495 0.74 HDAC2 (0.42) HDAC2HDAC8HDAC6PDGFRBPDGFRA
SCHEMBL22534215 0.71 APP (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111793025-B Method for modifying amino in molecule by oxazoline quaternary ammonium salt and application thereof 中国科学院上海药物研究所 2022-09-23 CN disclosed
CN-111793025-A Method for modifying amino in molecule by oxazoline quaternary ammonium salt and application thereof 中国科学院上海药物研究所 2020-10-20 CN disclosed