SCHEMBL28478249

SCHEMBL28478249

COc1ccc(Nc2nc3ccccc3c(C)c2C)cc1OC

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 17/20 0.65
ABCB1 P08183 10/20 0.65
ABCC1 P33527 6/20 0.65
MEN1 O00255 1/20 0.59
LMNA P02545 1/20 0.59
TP53 P04637 1/20 0.59
POLB P06746 1/20 0.59
MAPT P10636 1/20 0.59
KMT2A Q03164 1/20 0.59
GAA P10253 1/20 0.54
GFER P55789 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28469756 0.86 POLB (0.67) ABCG2ABCB1ABCC1MEN1LMNA
SCHEMBL2256504 0.84 ABCG2 (0.73) ABCG2ABCB1ABCC1MEN1LMNA
SCHEMBL14323064 0.81 ABCG2 (0.56) ABCG2ABCB1ABCC1MEN1LMNA
SCHEMBL3112389 0.80 ABCG2 (0.71) ABCG2ABCB1ABCC1MEN1LMNA
SCHEMBL22273241 0.79 ABCG2 (1.00) ABCG2ABCB1ABCC1MEN1LMNA
SCHEMBL8899168 0.79 ABCG2 (0.72) ABCG2ABCB1ABCC1MEN1LMNA
SCHEMBL7696554 0.79 ABCG2 (0.58) ABCG2ABCB1ABCC1MEN1LMNA
SCHEMBL28481400 0.78 NPY5R (0.63) ABCG2MEN1LMNATP53POLB
Hydrochloric Acid SCHEMBL8907536 0.78 ABCG2 (0.70) ABCG2ABCB1ABCC1MEN1LMNA
SCHEMBL13632592 0.78 TP53 (0.59) ABCG2ABCB1ABCC1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116143693-A 2-methylquinoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2023-05-23 CN claimed
CN-111825610-A 2-methylquinoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2020-10-27 CN claimed
CN-116143693-A 2-methylquinoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2023-05-23 CN disclosed
CN-111825610-B 2-methylquinoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2023-03-31 CN disclosed
CN-111825610-A 2-methylquinoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2020-10-27 CN disclosed