SCHEMBL28480249

SCHEMBL28480249

[CH2]c1nc2c(N)nc3cc(-c4cc[nH]n4)sc3c2n1Cc1ccc(OC)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 12/20 0.43
TLR8 Q9NR97 6/20 0.40
TYMS P04818 1/20 0.38
NPC1 O15118 2/20 0.35
PKM P14618 2/20 0.35
RAB9A P51151 2/20 0.35
KDM4E B2RXH2 2/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
DCTPP1 Q9H773 2/20 0.34
MAPT P10636 1/20 0.33
PDE8B O95263 1/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30598796 0.83 MEN1 (0.42) TLR7TYMSNPC1PKMRAB9A
SCHEMBL28473636 0.82 TLR7 (0.44) TLR7TLR8TYMSKDM4EKMT2A
SCHEMBL21566254 0.82 TLR7 (0.51) TLR7TLR8
SCHEMBL30598830 0.82 TLR7 (0.51) TLR7TLR8
SCHEMBL21550351 0.81 TLR7 (0.45) TLR7TLR8
SCHEMBL28476765 0.80 TLR7 (0.54) TLR7TLR8
SCHEMBL30598833 0.80 TLR7 (0.54) TLR7TLR8
SCHEMBL28468833 0.80 TLR7 (0.34) TLR7TLR8
SCHEMBL21566403 0.79 TLR7 (0.47) TLR7TLR8
SCHEMBL28472735 0.78 TLR7 (0.58) TLR7TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117263952-A Condensed-cyclic compound, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-12-22 CN disclosed
CN-111836814-B Condensed-cyclic compound, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-10-20 CN disclosed
CN-111836814-A Fused ring compound, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2020-10-27 CN disclosed