SCHEMBL28480388

SCHEMBL28480388

CC(C)C[C@](C)(N)COc1ccc(-c2cnnc(OC(=O)N(C)C(=O)OC(C)(C)C)c2)cc1C#N

nearest known ligand 0.63

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 20/20 0.63
CYP3A4 P08684 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28480652 0.88 AAK1 (0.52) AAK1CYP3A4
SCHEMBL28479890 0.87 AAK1 (0.70) AAK1CYP3A4
SCHEMBL28479886 0.87 AAK1 (0.70) AAK1CYP3A4
SCHEMBL28487584 0.85 AAK1 (0.72) AAK1CYP3A4
SCHEMBL28480390 0.83 AAK1 (0.67) AAK1CYP3A4
SCHEMBL28484964 0.82 AAK1 (0.61) AAK1CYP3A4
SCHEMBL20574090 0.80 AAK1 (0.68) AAK1CYP3A4
SCHEMBL20574095 0.80 AAK1 (0.68) AAK1CYP3A4
SCHEMBL20446849 0.78 AAK1 (0.85) AAK1CYP3A4
SCHEMBL28485418 0.77 AAK1 (0.63) AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112142655-A Biaryl kinase inhibitors 百时美施贵宝公司 2020-12-29 CN disclosed
CN-108368084-B Biaryl kinase inhibitors 百时美施贵宝公司 2020-10-16 CN disclosed