SCHEMBL28482114

SCHEMBL28482114

COc1ccc(C(C)c2nnc(-c3ccc(NC(=O)Nc4cccc(OC)c4)cc3)n2Cc2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.51
TP53 P04637 1/20 0.51
KDR P35968 2/20 0.48
KMT2A Q03164 3/20 0.47
PTGER3 P43115 3/20 0.47
MEN1 O00255 2/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 1/20 0.47
HIF1A Q16665 1/20 0.47
MAPT P10636 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
NTRK1 P04629 1/20 0.47
PDGFRB P09619 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
PDE6D O43924 1/20 0.46
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28482112 0.83 PDE6D (0.60) TSHRTP53KDRKMT2APTGER3
SCHEMBL28483909 0.81 KMT2A (0.52) TSHRTP53KMT2AMEN1KDM4E
SCHEMBL28478382 0.81 PDE6D (0.51) TSHRTP53KMT2AMEN1ALDH1A1
SCHEMBL28489680 0.77 SMN1; SMN2 (0.49) TP53KMT2AMEN1KDM4EALDH1A1
SCHEMBL28478423 0.76 PDE6D (0.57) KMT2AMEN1ALDH1A1HIF1ANTRK1
SCHEMBL28489558 0.73 PDE1A (0.43) TP53KMT2AMEN1KDM4EALDH1A1
SCHEMBL4117916 0.70 TP53 (0.76) TSHRTP53KMT2AMEN1ALDH1A1
SCHEMBL14442613 0.70 TP53 (0.84) TSHRTP53KMT2AMEN1ALDH1A1
SCHEMBL21295338 0.69 TP53 (0.83) TSHRTP53KMT2AMEN1ALDH1A1
SCHEMBL4105995 0.68 TP53 (0.81) TSHRTP53KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111875583-B Triazole derivative and preparation method and application thereof 中国科学院上海药物研究所 2021-06-15 CN disclosed
CN-109666022-B Triazole derivative and preparation method and application thereof 中国科学院上海药物研究所 2021-06-15 CN disclosed
CN-111875583-A Triazole derivative and preparation method and application thereof 中国科学院上海药物研究所 2020-11-03 CN disclosed