SCHEMBL28485950

SCHEMBL28485950

COC(=O)c1nc(C(C)(C)C)nn1Cc1c(C)cc(C)cc1C

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.40
TP53 P04637 2/20 0.38
SLC22A12 Q96S37 1/20 0.37
GAA P10253 2/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 4/20 0.32
MEN1 O00255 3/20 0.32
ALDH1A1 P00352 4/20 0.32
GLA P06280 1/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
KDM4E B2RXH2 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
EPHX2 P34913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17647954 0.89 SLC22A12 (0.37) MAPTSLC22A12KMT2AALDH1A1HTT
SCHEMBL17658947 0.86 SLC22A12 (0.42) TP53SLC22A12KMT2AMEN1ALDH1A1
SCHEMBL28483273 0.85 SLC22A12 (0.41) TP53SLC22A12KMT2AMEN1ALDH1A1
Lithium Ion SCHEMBL17648309 0.84 SLC22A12 (0.38) MAPTSLC22A12CYP11B1CYP11B2
SCHEMBL17647244 0.73 MAPT (0.38) MAPTTP53SLC22A12GAARAB9A
SCHEMBL17649180 0.72 PTGS1 (0.34)
SCHEMBL17646963 0.71 MAPT (0.48) MAPTTP53SLC22A12GAARAB9A
SCHEMBL2871405 0.68 MAPK1 (0.53) MAPTGAAALDH1A1LMNAKDM4E
SCHEMBL17648044 0.67 SLC22A12 (0.39) MAPTSLC22A12KMT2AMEN1ALDH1A1
SCHEMBL17648305 0.66 GRN (0.63) MAPTSLC22A12GAAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107690281-B Cystic fibrosis transmembrane transduction modulator modulators 弗特克斯药品有限公司 2020-11-17 CN disclosed