SCHEMBL28488268

SCHEMBL28488268

C[C@@H](NC(=O)OC(C)(C)C)C(=O)NCCCNC1CCCc2c1[nH]c1ccc(Br)cc21

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.47
KCNH2 Q12809 1/20 0.47
BRD3 Q15059 7/20 0.47
GAA P10253 1/20 0.46
CASP6 P55212 1/20 0.46
PRMT5 O14744 2/20 0.44
CDC42 P60953 1/20 0.43
DHODH Q02127 1/20 0.40
PARP1 P09874 1/20 0.39
AAK1 Q2M2I8 1/20 0.39
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28494320 0.92 CYP2D6 (0.46) CYP2D6KCNH2BRD3GAACASP6
SCHEMBL28494318 0.92 CYP2D6 (0.46) CYP2D6KCNH2BRD3GAACASP6
SCHEMBL20615752 0.90 BRD3 (0.52) CYP2D6KCNH2BRD3GAACASP6
SCHEMBL22529416 0.88 BRD3 (0.49) CYP2D6KCNH2BRD3GAACASP6
SCHEMBL30787992 0.88 BRD3 (0.49) CYP2D6KCNH2BRD3GAACASP6
SCHEMBL28488714 0.86 BRD3 (0.49) CYP2D6KCNH2BRD3GAACASP6
SCHEMBL20615443 0.86 BRD3 (0.55) CYP2D6KCNH2BRD3GAACASP6
SCHEMBL30787999 0.86 BRD3 (0.47) CYP2D6KCNH2BRD3GAACASP6
SCHEMBL30787997 0.86 BRD3 (0.47) CYP2D6KCNH2BRD3GAACASP6
SCHEMBL28498110 0.84 CYP2D6 (0.54) CYP2D6KCNH2BRD3GAACASP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107739371-B Tetrahydrocarbazole micromolecule organic compound, application thereof in preparing antibacterial drugs and preparation method thereof 华东师范大学 2020-08-25 CN disclosed