SCHEMBL28488685

SCHEMBL28488685

C=C(OCCC)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)OC(C)(C)C)CC4)cn3)nc2n(C2CCCC2)c1=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.67
CDK6 Q00534 8/20 0.67
CDK12 Q9NYV4 1/20 0.64
CCND1 P24385 13/20 0.63
CCND3 P30281 12/20 0.63
CCND2 P30279 11/20 0.63
CDK2 P24941 3/20 0.63
CCNA2 P20248 2/20 0.63
CDK9 P50750 2/20 0.63
CHEK1 O14757 1/20 0.59
DAPK3 O43293 1/20 0.59
CCNT1 O60563 1/20 0.59
CCNT2 O60583 1/20 0.59
ROCK2 O75116 1/20 0.59
STK16 O75716 1/20 0.59
CCNK O75909 1/20 0.59
PDE5A O76074 1/20 0.59
PRKD3 O94806 1/20 0.59
CCNB2 O95067 1/20 0.59
ABCB11 O95342 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29600291 0.96 CDK4 (0.66) CDK4CDK6CDK12CCND1CCND3
SCHEMBL2076205 0.96 CDK4 (0.66) CDK4CDK6CDK12CCND1CCND3
SCHEMBL2077623 0.95 CDK4 (0.70) CDK4CDK6CDK12CCND1CCND3
SCHEMBL4832945 0.94 CDK4 (0.67) CDK4CDK6CDK12CCND1CCND3
SCHEMBL29507410 0.90 CDK4 (0.77) CDK4CDK6CDK12CCND1CCND3
SCHEMBL4442470 0.90 CDK4 (0.77) CDK4CDK6CDK12CCND1CCND3
SCHEMBL30643549 0.90 CDK4 (0.62) CDK4CDK6CDK12CCND1CCND3
SCHEMBL17550859 0.89 CDK4 (0.68) CDK4CDK6CDK12CCND1CCND3
SCHEMBL17311359 0.89 CDK4 (0.72) CDK4CDK6CDK12CCND1CCND3
SCHEMBL29564471 0.89 CDK4 (0.80) CDK4CDK6CDK12CCND1CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111892590-A New piparib new intermediate, crystal form and preparation method thereof 齐鲁制药有限公司 2020-11-06 CN claimed
CN-111892590-A New piparib new intermediate, crystal form and preparation method thereof 齐鲁制药有限公司 2020-11-06 CN disclosed
CN-111892590-A New piparib new intermediate, crystal form and preparation method thereof 齐鲁制药有限公司 2020-11-06 CN disclosed