SCHEMBL28488693

SCHEMBL28488693

COc1cc2nccc(Oc3ccc(N(C(=O)C4(C(N)=O)CC4)C4CC4)c(Cl)c3)c2cc1C(N)=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.61
RET P07949 8/20 0.61
PDGFRB P09619 3/20 0.61
PDGFRA P16234 3/20 0.61
KIT P10721 2/20 0.61
FGFR1 P11362 2/20 0.61
FLT1 P17948 2/20 0.61
FLT4 P35916 2/20 0.61
EGFR P00533 1/20 0.61
AURKB Q96GD4 5/20 0.59
ABL1 P00519 2/20 0.59
RIPK2 O43353 1/20 0.59
ERN1 O75460 1/20 0.59
STK10 O94804 1/20 0.59
MAP3K6 O95382 1/20 0.59
ESR1 P03372 1/20 0.59
ADORA3 P0DMS8 1/20 0.59
BCR P11274 1/20 0.59
NQO2 P16083 1/20 0.59
TBXA2R P21731 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28499127 0.92 AXL (0.55) KDRRETPDGFRBPDGFRAKIT
SCHEMBL28490999 0.91 KDR (0.52) KDRRETPDGFRBPDGFRAKIT
SCHEMBL30148083 0.90 KDR (0.64) KDRRETPDGFRBPDGFRAKIT
SCHEMBL2721687 0.90 KDR (0.64) KDRRETPDGFRBPDGFRAKIT
SCHEMBL28492056 0.88 AXL (0.55) KDRRETPDGFRBPDGFRAKIT
SCHEMBL29729418 0.86 AXL (0.54) KDRRETPDGFRBPDGFRAKIT
SCHEMBL28796986 0.86 AXL (0.54) KDRRETPDGFRBPDGFRAKIT
SCHEMBL28491003 0.85 KDR (0.52) KDRRETPDGFRBPDGFRAKIT
SCHEMBL29729490 0.85 KDR (0.52) KDRRETPDGFRBPDGFRAKIT
SCHEMBL29729435 0.83 AXL (0.55) KDRRETPDGFRBPDGFRAKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111892536-B Substituted quinoline carboxamides and their use 北京福元医药股份有限公司 2022-06-28 CN disclosed
CN-111892536-A Substituted quinoline carboxamides and their use 北京福元医药股份有限公司 2020-11-06 CN disclosed