SCHEMBL28490

SCHEMBL28490

Cc1c(C)c(N)c2c(N)ccc(C)c2c1C

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.39
CYP3A4 P08684 6/20 0.34
ALDH1A1 P00352 4/20 0.34
TDP1 Q9NUW8 4/20 0.34
TSHR P16473 3/20 0.34
CD44 P16070 1/20 0.34
CASP1 P29466 1/20 0.34
PIK3CA P42336 1/20 0.33
KDM4E B2RXH2 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TP53 P04637 1/20 0.31
THRB P10828 1/20 0.31
ALOX15 P16050 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29712483 1.00 POLB (0.39) POLBCYP3A4ALDH1A1TDP1TSHR
SCHEMBL4657946 0.77 CYP3A4 (0.46) POLBCYP3A4ALDH1A1TDP1TSHR
SCHEMBL25144754 0.75 CYP3A4 (0.43) POLBCYP3A4ALDH1A1TDP1TSHR
SCHEMBL11815258 0.75 CYP3A4 (0.43) POLBCYP3A4ALDH1A1TDP1TSHR
SCHEMBL20380560 0.75 CYP3A4 (0.43) POLBCYP3A4ALDH1A1TDP1TSHR
SCHEMBL9223063 0.73 POLB (0.44) POLBCYP3A4ALDH1A1TDP1TSHR
SCHEMBL11504041 0.70 CD44 (0.36) POLBCYP3A4ALDH1A1TDP1TSHR
SCHEMBL23457967 0.70 POLB (0.41) POLBCYP3A4ALDH1A1TDP1TSHR
SCHEMBL9378000 0.69 HPGD (0.32) CYP3A4ALDH1A1TSHRCASP1KDM4E
SCHEMBL16132694 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 296 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250135721-A1 STEREOLITHOGRAPHY THREE-DIMENSIONAL PRINTING OF FOAM MATERIALS CONTAINING HOLLOW MICROSPHERES IMPRESSIO INC. (US) 2025-05-01 US claimed
WO-2023150160-A1 STEREOLITHOGRAPHY THREE-DIMENSIONAL PRINTING OF FOAM MATERIALS CONTAINING HOLLOW MICROSPHERES IMPRESSIO INC. (US) 2023-08-10 WO claimed
EP-4041218-A1 PROCESS FOR PREPARATION OF DIROXIMEL FUMARATE Glenmark Life Sciences Limited (IN) 2022-08-17 EP claimed
WO-2021053476-A1 PROCESS FOR PREPARATION OF DIROXIMEL FUMARATE GLENMARK LIFE SCIENCES LIMITED (IN) 2021-03-25 WO claimed
CN-105642136-B One kind containing soft segment and hard section copolymer ammonium cross-linking type anion-exchange membrane and preparation method thereof 北京化工大学 2018-07-27 CN claimed
CN-106398080-A Aminated cross-linked segmented copolymer/graphene composite material and preparation method thereof 北京化工大学 2017-02-15 CN claimed
CN-105669882-A Azonium-ionized poly(styrene-b-isobutylene-b-styrene) triblock copolymer and preparation method thereof 北京化工大学 2016-06-15 CN claimed
EP-2938712-A1 ULTRA-LOW SAPS LUBRICANTS FOR INTERNAL COMBUSTION ENGINES Chevron Oronite Company LLC (US) 2015-11-04 EP claimed
EP-2938713-A2 ULTRA-LOW SAPS LUBRICANTS FOR INTERNAL COMBUSTION ENGINES Chevron Oronite Company LLC (US) 2015-11-04 EP claimed
WO-2014105311-A2 ULTRA-LOW SAPS LUBRICANTS FOR INTERNAL COMBUSTION ENGINES CHEVRON ORONITE COMPANY LLC (US) 2014-07-03 WO claimed
WO-2014105312-A1 ULTRA-LOW SAPS LUBRICANTS FOR INTERNAL COMBUSTION ENGINES CHEVRON ORONITE COMPANY LLC (US) 2014-07-03 WO claimed
CN-101687120-B Method for direct elution of reactive18F fluoride ions from anion exchange resins in an organic medium suitable for radiolabelling, without any evaporation step, by using strong organic bases TRASIS S A 2013-12-18 CN claimed
EP-1942949-A1 METHOD FOR THE SYNTHESIS OF PENTAPENDANT ENANTIOMER-PURE CHELATORS AND PROCESS FOR THERAPEUTICALLY ACTIVE BIO-CONJUGATES PREPARATION BY A COVALENT BINDING OF THEREOF Therapharm GmbH (CH) 2008-07-16 EP claimed
WO-2007028639-A1 METHOD FOR THE SYNTHESIS OF PENTAPENDANT ENANTIOMER-PURE CHELATORS AND PROCESS FOR THERAPEUTICALLY ACTIVE BIO-CONJUGATES PREPARATION BY A COVALENT BINDING OF THEREOF THERAPHARM GMBH (CH) 2007-03-15 WO claimed
EP-0415030-A2 1-Substituted-1,2-dihydro-4-[(substituted)-phenyl]imidazo-[1,5-A]pyrimidine-8-carbonitriles AMERICAN CYANAMID COMPANY (US) 1991-03-06 EP claimed
EP-4626546-A1 HETEROCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2025-10-08 EP disclosed
EP-4587445-A1 IMPROVED METHODS FOR PREPARING N-METHYL ALANINE ESTERS OF MAYTANSINOL ImmunoGen, Inc. (US) 2025-07-23 EP disclosed
EP-0264773-A1 4,5-dihydro and 4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidines AMERICAN CYANAMID COMPANY (US) 1988-04-27 EP disclosed
EP-0219876-A2 Antihypertensive agents comprising 2-alkynyladenosines as active ingredients Yamasa Shoyu Kabushiki Kaisha (JP) 1987-04-29 EP disclosed
US-4036863-A Trinapthylmethane compounds POLAROID CORPORATION (US) 1977-07-19 US disclosed