SCHEMBL28495249

SCHEMBL28495249

Clc1ncnc2cnc(OCCN3CCOCC3)cc12

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
SIGMAR1 Q99720 8/20 0.45
TSHR P16473 1/20 0.44
KCNH2 Q12809 1/20 0.43
KDR P35968 2/20 0.43
EPHA2 P29317 1/20 0.43
EPHB4 P54760 1/20 0.43
NPC1 O15118 1/20 0.43
EGFR P00533 2/20 0.41
FGFR1 P11362 1/20 0.41
FLT1 P17948 1/20 0.41
FLT4 P35916 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28487050 0.79 KDR (0.52) KDM4ETSHRKDREPHA2EPHB4
SCHEMBL6368598 0.78 IRAK4 (0.48) SIGMAR1EGFR
SCHEMBL4507750 0.78 KDM4E (0.61) KDM4EALDH1A1SIGMAR1TSHRKDR
SCHEMBL3425922 0.78 KDR (0.67) KDM4EKCNH2KDREPHA2EPHB4
SCHEMBL1011324 0.78 KDR (0.67) KDM4EKCNH2KDREPHA2EPHB4
SCHEMBL3205812 0.78 KDM4E (0.52) KDM4EALDH1A1SIGMAR1TSHRKCNH2
SCHEMBL25286424 0.78 CYP1A2 (0.49) KDM4EALDH1A1TSHRKDREPHA2
SCHEMBL4985461 0.75 KDR (0.58) KDREPHA2EPHB4EGFRFGFR1
SCHEMBL18256900 0.75 KDM4E (0.50) KDM4EALDH1A1SIGMAR1TSHRKCNH2
SCHEMBL13503071 0.73 EGFR (0.56) KDM4EKCNH2KDREPHB4EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108341813-B Substituted 1- (isoxazol-3-yl) -3- (3-fluoro-4-phenyl) urea derivative and preparation method and application thereof 四川大学 2020-11-17 CN disclosed