SCHEMBL28495356

SCHEMBL28495356

COC(=O)c1nc(OC)c(Br)cc1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.42
KDM4E B2RXH2 6/20 0.40
CFTR P13569 6/20 0.40
ALDH1A1 P00352 4/20 0.39
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PKM P14618 3/20 0.38
MAPK8 P45983 1/20 0.37
MAPK9 P45984 1/20 0.37
GAA P10253 3/20 0.36
HSD17B10 Q99714 3/20 0.36
HPGD P15428 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GLA P06280 1/20 0.36
MAPT P10636 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
ATM Q13315 1/20 0.36
RCE1 Q9Y256 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28491736 0.85 POLB (0.44) KDM4ECFTRALDH1A1POLBL3MBTL1
SCHEMBL20745291 0.85 HSD17B10 (0.40) KDM4ECFTRALDH1A1POLBL3MBTL1
SCHEMBL25359695 0.83 NPSR1 (0.45) NPSR1KDM4ECFTRALDH1A1PKM
SCHEMBL30475032 0.82 NPSR1 (0.44) NPSR1KDM4ECFTRALDH1A1L3MBTL1
SCHEMBL25305744 0.82 NPSR1 (0.44) NPSR1KDM4ECFTRALDH1A1L3MBTL1
SCHEMBL23364116 0.81 GAA (0.46) NPSR1KDM4ECFTRALDH1A1L3MBTL1
SCHEMBL25096003 0.81 NPSR1 (0.42) NPSR1KDM4ECFTRALDH1A1L3MBTL1
SCHEMBL30218091 0.81 NPSR1 (0.42) NPSR1KDM4ECFTRALDH1A1L3MBTL1
SCHEMBL25360368 0.77 KDM4E (0.44) KDM4ECFTRALDH1A1POLBL3MBTL1
SCHEMBL29824155 0.77 KDM4E (0.44) KDM4ECFTRALDH1A1POLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112110918-B Spiro substituted pyrimido cyclic compounds, process for their preparation and their use in medicine 劲方医药科技(上海)有限公司 2023-08-22 CN disclosed
CN-112110918-A Spiro-substituted pyrimido-cyclic compounds, preparation method and medical application thereof 劲方医药科技(上海)有限公司 2020-12-22 CN disclosed