SCHEMBL28501194

SCHEMBL28501194

Cc1ccc2c(cnn2C2CCCCO2)c1C1Cc2ncnc(N3CCN(C(=O)CC(C)N(C)C(=O)OC(C)(C)C)CC3)c2CC1C

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KRAS P01116 3/20 0.44
AKT1 P31749 8/20 0.32
KIT P10721 2/20 0.32
ATR Q13535 3/20 0.31
AKT2 P31751 5/20 0.31
AKT3 Q9Y243 5/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21733504 0.85 KRAS (0.48) KRASKITATR
SCHEMBL21722284 0.82 KRAS (0.65) KRAS
SCHEMBL21722208 0.80 KRAS (0.48) KRASATR
SCHEMBL21243885 0.77 KRAS (0.41) KRASKITATR
SCHEMBL21243891 0.76 KIT (0.39) KRASKIT
SCHEMBL21243944 0.75 KRAS (0.48) KRASKITATR
SCHEMBL21722212 0.75 KRAS (0.40) KRASKITATR
SCHEMBL21733530 0.75 KRAS (0.39) KRASKITATR
SCHEMBL21722422 0.75 KRAS (0.60) KRAS
SCHEMBL21733673 0.71 KRAS (0.52) KRASAKT1AKT2AKT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112119075-B Condensed ring compound 豪夫迈·罗氏有限公司 2024-03-12 CN disclosed
CN-112119075-A Fused ring compound 豪夫迈·罗氏有限公司 2020-12-22 CN disclosed