SCHEMBL28501362

SCHEMBL28501362

COC(=O)c1n[nH]c2cc(Br)cc(F)c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
STAT3 P40763 1/20 0.46
HIF1A Q16665 1/20 0.46
KDM4C Q9H3R0 1/20 0.40
ALPL P05186 3/20 0.39
LRRK2 Q5S007 1/20 0.38
MAP2K4 P45985 1/20 0.38
MAPK1 P28482 1/20 0.36
NOTUM Q6P988 1/20 0.36
DYRK1A Q13627 1/20 0.36
GPR17 Q13304 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
MAPK10 P53779 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
FLT3 P36888 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
MMP8 P22894 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23872474 0.85 KDM4E (0.48) KDM4ESTAT3HIF1AKDM4CALPL
SCHEMBL28496732 0.82 GPR17 (0.45) DYRK1AGPR17IDO1PRKAB2PRKAG1
SCHEMBL31647132 0.77 KDM4E (0.46) KDM4ESTAT3HIF1AKDM4CALPL
SCHEMBL2862825 0.77 KDM4E (0.59) KDM4ESTAT3HIF1AKDM4CALPL
SCHEMBL31725399 0.74 KDM4E (0.52) KDM4ESTAT3HIF1AKDM4CALPL
SCHEMBL13132306 0.74 MAP2K4 (0.43) KDM4ESTAT3HIF1AALPLMAP2K4
SCHEMBL30258217 0.74 KDM4E (0.63) KDM4ESTAT3HIF1AMAP2K4DYRK1A
SCHEMBL498163 0.74 KDM4E (0.63) KDM4ESTAT3HIF1AMAP2K4DYRK1A
SCHEMBL2599805 0.72 KDM4E (0.60) KDM4ESTAT3HIF1AKDM4CLRRK2
SCHEMBL31162464 0.72 PDPK1 (0.34) MAPK1DYRK1AGPR17RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111995577-A Synthetic method of 4-fluoro indazole 3-carbonitrile or derivatives thereof 上海代为化学科技有限公司 2020-11-27 CN disclosed