SCHEMBL28503202

SCHEMBL28503202

Clc1c[c]ccc1-c1cncc(Br)c1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.39
CYP11B2 P19099 3/20 0.37
CYP11B1 P15538 2/20 0.37
PTK2 Q05397 1/20 0.35
P4HTM Q9NXG6 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771 0.76 CYP2A6 (0.47) CYP2A6PTK2KMT2A
SCHEMBL28822926 0.75 MAPK1 (0.33) CYP2A6KMT2A
SCHEMBL5110030 0.75 AHR (0.48) CYP2A6PTK2KMT2A
SCHEMBL2155431 0.73 CYP2A6 (0.52) CYP2A6CYP11B2CYP11B1PTK2HDAC6
SCHEMBL5888962 0.72 CYP2A6 (0.40) CYP2A6CYP11B2CYP11B1PTK2KMT2A
SCHEMBL27893679 0.71 CYP2A6 (0.46) CYP2A6CYP11B2CYP11B1PTK2KMT2A
SCHEMBL28514778 0.71 PDGFRB (0.34)
SCHEMBL28906118 0.71
SCHEMBL28504316 0.70 CYP11B1 (0.34) CYP11B2CYP11B1
SCHEMBL1135190 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243374-A SREBP inhibitors comprising a 6-membered central ring 卡普勒斯疗法有限责任公司 2021-01-19 CN disclosed