SCHEMBL28512205

SCHEMBL28512205

CCOC(=O)c1cccc2c1CN(c1nc3c([nH]1)CCC(C(F)(F)F)C3)C2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC11 Q96DB2 6/20 0.45
USP2 O75604 2/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
RXFP1 Q9HBX9 1/20 0.34
LMNA P02545 1/20 0.34
PRKD3 O94806 1/20 0.34
MAP4K4 O95819 1/20 0.34
PIM1 P11309 1/20 0.34
CLK2 P49760 1/20 0.34
MAP4K2 Q12851 1/20 0.34
CAMK2D Q13557 1/20 0.34
DYRK1A Q13627 1/20 0.34
PIM3 Q86V86 1/20 0.34
AURKB Q96GD4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30039897 1.00 HDAC11 (0.45) HDAC11USP2MEN1ALDH1A1POLB
SCHEMBL30039180 1.00 HDAC11 (0.45) HDAC11USP2MEN1ALDH1A1POLB
SCHEMBL21496820 0.91 HDAC11 (0.49) HDAC11C5AR1TIPARPHDAC6
SCHEMBL25932035 0.88 HDAC11 (0.47) HDAC11USP2MEN1ALDH1A1POLB
SCHEMBL25932026 0.88 HDAC11 (0.47) HDAC11USP2MEN1ALDH1A1POLB
SCHEMBL21496749 0.86 HDAC11 (0.47) HDAC11TIPARPSPRHDAC6
SCHEMBL28518722 0.86 HDAC11 (0.47) HDAC11TIPARPSPRHDAC6
SCHEMBL28521107 0.86 HDAC11 (0.47) HDAC11TIPARPSPRHDAC6
SCHEMBL21496744 0.84 HDAC11 (0.61) HDAC11TIPARPHDAC6
SCHEMBL21500463 0.84 HDAC11 (0.61) HDAC11TIPARPHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112292370-A Isoindolines as HDAC inhibitors 瓦洛早期发现股份有限公司 2021-01-29 CN disclosed