SCHEMBL28512440

SCHEMBL28512440

NC(=O)C(C(N)=O)c1ccc([N+](=O)[O-])c(C(F)(F)F)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM8 O00222 2/20 0.53
GRM6 O15303 2/20 0.53
GRM4 Q14833 2/20 0.53
AR P10275 7/20 0.52
CYP3A4 P08684 3/20 0.52
LMNA P02545 2/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2C9 P11712 2/20 0.52
TSHR P16473 2/20 0.52
CYP2C19 P33261 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
CES2 O00748 1/20 0.52
ABCB11 O95342 1/20 0.52
ALDH1A1 P00352 1/20 0.52
GLA P06280 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
CHRM1 P11229 1/20 0.52
ALOX15 P16050 1/20 0.52
TBXA2R P21731 1/20 0.52
AADAC P22760 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3964971 0.88 GRM8 (0.56) GRM8GRM6GRM4ARCYP3A4
SCHEMBL3964959 0.88 GRM8 (0.56) GRM8GRM6GRM4ARCYP3A4
SCHEMBL9727361 0.87 AR (0.55) GRM8GRM6GRM4ARCYP3A4
SCHEMBL2746779 0.81 AR (0.49) GRM8GRM6GRM4ARCYP3A4
SCHEMBL10629315 0.80 AR (0.56) GRM8GRM6GRM4ARCYP3A4
SCHEMBL5842211 0.79 AR (0.50) GRM8GRM6GRM4ARCYP3A4
SCHEMBL2973491 0.78 PARP1 (0.55) GRM8GRM6GRM4ARCYP3A4
SCHEMBL18528104 0.77 GRM8 (0.52) GRM8GRM6GRM4ARCYP3A4
SCHEMBL16952504 0.77 AR (0.53) GRM8GRM6GRM4ARCYP3A4
SCHEMBL16952607 0.77 GRM8 (0.48) GRM8GRM6GRM4ARCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026027-B Substituted malonamide compounds and their use as antibacterial agents 邱浩杰 2020-10-02 CN disclosed